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GSK1904529A Chemical Structure

GSK1904529A

Cat. No. :BCP01719CAS No. :1089283-49-7Purity:98%
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Synonyms GSK 1904529A;GSK-1904529A;GSK 4529
CAS Number 1089283-49-7
Purity 98%
M. Wt 851.96
Formula C44H47F2N9O5S
Storage Store at -20°C
GSK1904529A is a reversible, ATP-competitive inhibitor and has enzyme-inhibitor binding values against IGF-1R and IR with Ki of 1.6 nM and 1.3 nM, respectively. GSK1904529A potently inhibits the ligand-induced phosphorylation of IGF-1R and IR at concentrations above 0.01 μM, followed by blocking downstream signaling (AKT, IRS-1, and ERK). GSK1904529A potently inhibits NIH-3T3/LISN, TC-71, SK-N-MC, SK-ES RD-ES cells with IC50 of 60 nM, 35 nM, 43 nM, 61 nM and 62 nM, respectively. GSK1904529A also

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