Encequidar mesylate New
Data Sheet
For research use only. Not for human use.
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| CAS No. | 849675-87-2 | Cat. No. | BCP33772 |
| Related Products | 2097125-58-9（Encequidar mesylate monohydrate） 849675-66-7（Encequidar） | ||
| Name | Encequidar mesylate | ||
| Synonyms | HM-30181 mesylate;HM30181 mesylate;HM 30181 mesylate; HM30181A mesylate; | ||
| SMILES | COC1=C(C=C2CN(CCC2=C1)CCC3=CC=C(C=C3)N4N=C(N=N4)C5=CC(=C(C=C5NC(=O)C6=CC(=O)C7=CC=CC=C7O6)OC)OC)OC.CS(=O)(=O)O | ||
| Chemical Name | |||
| Formula | C39H40N6O10S | M. Wt | 784.83 |
| Purity | 98% | Storage | Store at 4-8°C |
| Description | Encequidar is an oral P-glycoprotein (P-gp) inhibitor developed to enhance the oral bioavailability of P-gp substrate drugs. HM30181 showed the highest potency (IC(50)=0.63nM) among several MDR1 inhibitors, including cycloporin A, XR9576, and GF120918, and effectively blocked transepithelial transport of paclitaxel in MDCK monolayers (IC(50)=35.4nM). HM30181 is currently under clinical trials. | ||
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