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5 HT Receptor/Serotonin Receptor

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5 HT Receptor/Serotonin Receptor

结构式 货号 产品名称 CAS号
Pimethixene 结构式
BCP43719 匹美噻吨 314-03-4
Pimethixene is antihistamine and anticholinergic of the thioxanthene chemical class that is often used to treat hyperactivity, anxiety, sleep disorders, and allergy. It is also used for anesthesia and as a bronchodilator (to dilate the bronchi and bronchioles for more airflow).
Pimethixene maleate 结构式
BCP43718 马来酸甲哌硫蒽 13187-06-9
Pimethixene maleate is antihistamine and antiserotonergic compound, acts as an antimigraine agent. Pimethixene maleate is a highly potent antagonist of 5-HT1A, 5-HT2A, 5-HT2B, 5-HT2C, histamine H1, dopamine D2 and D4.4 as well as muscarinic M1 and M2 receptors, with pKis of 7.63, 10.22, 10.44, 8.42, 10.14, 8.19, 7.54, 8.61 and 9.38, respectively.
SB 203186 hydrochloride 结构式
BCP42428 SB 203186盐酸盐 135938-17-9
SB203186 is potent 5-HT4 receptor antagonist with high affinity for human atrial 5-HT4 receptors.
Indophagolin 结构式
BCP41936 Indophagolin 1207660-00-1
Indophagolin is a potent autophagy inhibitor with and IC50 value of 140 nM. Indophagolin also shows activity on the purinergic receptors with IC50 values of 2.40 μM, 3.49 μM and 2.71 μM for the P2X1, P2X3 and P2X4 receptors, respectively.
Buspirone 结构式
BCP41132 丁螺环酮 36505-84-7
Buspirone is an anxiolytic psychotropic drug of the azapirone chemical class. It is primarily used to treat generalized anxiety disorder (GAD). Unlike most drugs predominantly used to treat anxiety, buspirone's pharmacology is not related to benzodiazepines or barbiturates, and so does not carry the risk of physical dependence and withdrawal symptoms for which those drug classes are known.
RS67333 结构式
BCP40415 RS67333 160845-95-4
RS-67333 is a 5-HT4R partial agonist that shows efficacy at 0.3 and 1.0 mg/kg, ip.
Tesofensine 结构式
BCP37838 特索芬辛 402856-42-2
Tesofensine, an azabicyclo compound, has been found to be a 5-HT receptor inhibitor and could be used in the treatment of obesity.
GR 125743 结构式
BCP37767 GR 125743 148547-33-5
GR 125743 is a novel 5-HT1B/1D receptor antagonist.
(S)-PF-04995274 结构式
BCP37093 (S)-PF-04995274 2170558-28-6
PF-04995274 is a 5-HT4 receptor partial agonist with Ki = 0.15 - 0.46 nM for 5-HT4 isoforms a, b, d and e, developed for the treatment of Alzheimer's disease (AD).
Org-12962 结构式
BCP37028 Org-12962 132834-56-1
Org-12962 is a 5-HT 2C receptor agonist potentially for the treatment of depression.
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