首页   >  
Neuro Signaling Pathway
  • GPCR/G Protein
  >  
Histamine Receptor

所有产品分类

所有产品

信号通路

研究领域

天然产物

抗体

多肽

催化剂

杂质对照品

医药中间体

基础原料

Histamine Receptor

结构式 货号 产品名称 CAS号
Terfenadine 结构式
BCP43974 特非那定 50679-08-8
Terfenadine is a potent open-channel blocker of hERG with a mean IC50 of 204 nM.
Pimethixene 结构式
BCP43719 匹美噻吨 314-03-4
Pimethixene is antihistamine and anticholinergic of the thioxanthene chemical class that is often used to treat hyperactivity, anxiety, sleep disorders, and allergy. It is also used for anesthesia and as a bronchodilator (to dilate the bronchi and bronchioles for more airflow).
Pimethixene maleate 结构式
BCP43718 马来酸甲哌硫蒽 13187-06-9
Pimethixene maleate is antihistamine and antiserotonergic compound, acts as an antimigraine agent. Pimethixene maleate is a highly potent antagonist of 5-HT1A, 5-HT2A, 5-HT2B, 5-HT2C, histamine H1, dopamine D2 and D4.4 as well as muscarinic M1 and M2 receptors, with pKis of 7.63, 10.22, 10.44, 8.42, 10.14, 8.19, 7.54, 8.61 and 9.38, respectively.
Chlorphenoxamine 结构式
BCP43687 氯苯沙明 77-38-3
Chlorphenoxamine is a diarylmethane. It has a role as an anticoronaviral agent.
Thioperamide 结构式
BCP39480 Thioperamide 106243-16-7
Thioperamide is a potent histamine H3 and H4 antagonist/inverse agonist (Ki = 25 and 27 nM for human recombinant H3 and H4 receptors, respectively). Thioperamide can cross the blood-brain barrier freely.
Thioperamide maleate 结构式
BCP39479 硫丙咪胺马来酸 148440-81-7
Thioperamide maleate is a selective histamine H3 receptor antagonist that crosses the blood-brain barrier.
JNJ-5207852 结构式
BCP37369 JNJ-5207852 398473-34-2
JNJ-5207852 is a selective and potent histamine H3 receptor (H3R) antagonist, with pKis of 8.9, 9.24 for rat and human H3R, respectively.
Thonzylamine 结构式
BCP25799 松齐拉敏 91-85-0
Thonzylamine is a first-generation ethylenediamine H1-antihistamine.
Doxepin-d3 Hydrochloride 结构式
BCP33258 盐酸多虑平D3 347840-07-7
Doxepin D3 Hydrochloride is a deuterium labeled Doxepin Hydrochloride.Doxepin is a tricyclic antidepressant (TCA) used for the treatment of major depression and anxiety.
Clobenpropit dihydrobromide 结构式
BCP33039 丙酸倍氯松二溴酸盐 145231-35-2
Clobenpropit dihydrobromide is an extremely potent histamine H3 antagonist/inverse agonist (pA2=9.93). Also displays partial agonist activity at H4 receptors; induces eosinophil shape change with an EC50 of 3 nM.
123下一页末页共 105 条记录 1 / 11 页 
2853530910