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Histamine Receptor

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Histamine Receptor

Chemical Structure Cat. No. Product Name CAS No.
Izuforant Chemical Structure
 BCP48744 Izuforant 1429374-83-3
Izuforant is an orally active histamine H4 receptor (H4R) antagonist. Izuforant also shows binding affinity of human serotonin 3 receptor (h5-HT3R). Izuforant exhibits strong anti-pruritic and anti-inflammatory efficacies.
JNJ 10191584 Chemical Structure
 BCP48111 JNJ 10191584 73903-17-0
JNJ-10191584 is a selective, orally active antagonist of the histamine H4 receptor.
JNJ 10191584 maleate Chemical Structure
 BCP48110 JNJ 10191584 maleate 869497-75-6
JNJ 10191584 maleate is a highly selective histamine H4 receptor silent antagonist.
GSK-239512 Chemical Structure
 BCP48003 GSK-239512 720691-69-0
GSK-239512 is a histamine H3 receptor antagonist.
Antazoline phosphate Chemical Structure
 BCP44465 Antazoline phosphate 154-68-7
Antazoline phosphate is an antihistamine with anticholinergic properties used to relieve nasal congestion and the symptoms of allergic conjunctivitis. Antazoline is an ethylenediamine derivative with histamine H1 antagonistic and sedative properties. Antazoline antagonizes histamine H1 receptor and prevents the typical allergic symptoms caused by histamine activities on capillaries, skin, mucous membranes, and gastrointestinal and bronchial smooth muscles.
Terfenadine Chemical Structure
 BCP43974 Terfenadine 50679-08-8
Terfenadine is a potent open-channel blocker of hERG with a mean IC50 of 204 nM.
Pimethixene Chemical Structure
 BCP43719 Pimethixene 314-03-4
Pimethixene is antihistamine and anticholinergic of the thioxanthene chemical class that is often used to treat hyperactivity, anxiety, sleep disorders, and allergy. It is also used for anesthesia and as a bronchodilator (to dilate the bronchi and bronchioles for more airflow).
Pimethixene maleate Chemical Structure
 BCP43718 Pimethixene maleate 13187-06-9
Pimethixene maleate is antihistamine and antiserotonergic compound, acts as an antimigraine agent. Pimethixene maleate is a highly potent antagonist of 5-HT1A, 5-HT2A, 5-HT2B, 5-HT2C, histamine H1, dopamine D2 and D4.4 as well as muscarinic M1 and M2 receptors, with pKis of 7.63, 10.22, 10.44, 8.42, 10.14, 8.19, 7.54, 8.61 and 9.38, respectively.
Thioperamide Chemical Structure
 BCP39480 Thioperamide 106243-16-7
Thioperamide is a potent histamine H3 and H4 antagonist/inverse agonist (Ki = 25 and 27 nM for human recombinant H3 and H4 receptors, respectively). Thioperamide can cross the blood-brain barrier freely.
Thioperamide maleate Chemical Structure
 BCP39479 Thioperamide maleate 148440-81-7
Thioperamide maleate is a selective histamine H3 receptor antagonist that crosses the blood-brain barrier.
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