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PPAR

结构式 货号 产品名称 CAS号
Saroglitazar magnesium 结构式
BCP49279 沙罗格列扎镁盐 1639792-20-3
Saroglitazar magnesium is a dual agonist at the PPARα and PPARγ of the peroxisome proliferator-activated receptor (PPAR).
Bocidelpar hemisulfate 结构式
BCP49259 Bocidelpar hemisulfate BH
Bocidelpar, also known as ASP0367 or MA-0211, is a peroxisome proliferator-activated receptor (PPAR) delta agonist.
Bocidelpar sulfate 结构式
BCP49258 Bocidelpar sulfate 2095128-21-3
Bocidelpar is a peroxisome proliferator-activated receptor (PPAR) delta agonist.
Mavodelpar sodium 结构式
BCP49236 Mavodelpar sodium 1604815-32-8
Mavodelpar is a selective PPARδ agonist.
Edaglitazone 结构式
BCP26908 依格列宗 213411-83-7
Edaglitazone is a PPARγ agonist potentially for the treatment of type 2 diabetes. Edarglitazone, restores acute inflammatory responses to cerebral hypoxia-ischemia in the diabetic ob/ob mouse.
PTGR2-IN-1 结构式
BCP48929 PTGR2-IN-1 349093-44-3
PTGR2-IN-1 is a potent PTGR2 inhibitor with an IC50 of ~0.7 μM.
Elafibranor 结构式
BCP31152 Elafibranor 824932-88-9
Elafibranor (GFT505) is an agonist of the peroxisome proliferator-activated receptor-α(PPAR-alpha) and peroxisome proliferator-activated receptor-δ(PPAR-δ). It improves insulin sensitivity, glucose homeostasis, and lipid metabolism and reduces inflammation.
Bocidelpar 结构式
BCP45760 Bocidelpar 2095128-20-2
Bocidelpar is a peroxisome proliferator-activated receptor (PPAR) delta agonist.
SR1664 结构式
BCP45759 SR1664 1338259-05-4
SR1664 is a potent and selective PPARγ inhibitor with potential antidiabetic activity.
AMG-131 结构式
BCP45654 AMG-131 315224-26-1
AMG-131 is a hypoglycemic agent. It is a potent PPARγ partial agonist that displays robust glucose-lowering activity in rodent models of diabetes while exhibiting a reduced side-effects profile compared to marketed TZDs.
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