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Protein Arginine Deiminase

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Protein Arginine Deiminase

Chemical Structure Cat. No. Product Name CAS No.
BMS-P5 hydrochloride Chemical Structure
BCP44953 BMS-P5 hydrochloride 1549811-36-0
BMS-P5 is a Novel Peptidylarginine Deiminase 4 (PAD4) Inhibitor with pIC50 values in the range of 5-​7.5.
Cl-amidine TFA Chemical Structure
BCP43968 Cl-amidine TFA 1043444-18-3
Cl-amidine is an irreversible pan-peptidylarginine deiminase (PAD) inhibitor with IC50 values of 5.9 ± 0.3 μM, 0.8 ± 0.3 μM, 6.2 ± 1.0 μM for PAD4, PAD1 and PAD3, respectively. Cl-amidine induces apoptosis.
GSK106 hydrochloride Chemical Structure
BCP37874 GSK106 hydrochloride 1652591-82-6
GSK106 is a negative control compound used in binding and functional assays for PAD4 inhibitors.
GSK121 trifluoroacetate salt Chemical Structure
BCP37872 GSK121 trifluoroacetate salt 1652591-80-4
GSK121 is a selective PAD4 inhibitor.
BMS-P5 Chemical Structure
BCP37124 BMS-P5 1550371-22-6
BMS-P5 free base is a specific and orally active peptidylarginine deiminase 4 (PAD4) inhibitor.
BB-Cl-Amidine hydrochloride Chemical Structure
BCP36632 BB-Cl-Amidine hydrochloride BB-Cl-AmidineHCl
BB-Cl-Amidine hydrochloride is a peptidylarginine deminase (PAD) inhibitor.
GSK199 hydrochloride Chemical Structure
BCP30343 GSK199 hydrochloride 1549811-53-1
GSK199 is a selective PAD4 inhibitor with half-maximum inhibitory concentration (IC50) values, in the absence of calcium, of 200 nM.
BB-Cl-Amidine Chemical Structure
BCP30300 BB-Cl-Amidine 1802637-39-3
BB-Cl-Amidine is a peptidylarginine deminase (PAD) inhibitor.
Cl-Amidine Chemical Structure
BCP20202 Cl-Amidine 913723-61-2
Cl-amidine is a peptidylarginine deminase (PAD) inhibitor, with an IC50 5.9±0.3 μM for PAD4.
GSK484 hydrochloride Chemical Structure
BCP25415 GSK484 hydrochloride 1652591-81-5
GSK484 hydrochloride is a specifc and reversible peptidyl arginine deiminase 4 (PAD4) inhibitor. It demonstrates high-affinity binding to PAD4 with IC50s of 50 nM in the absence of Calcium.
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