PNU-282987 S enantiomer free base

Description	PNU-282987 is a highly selective α7 nAChR agonist (Ki = 26 nM) displaying negligible blockade of α1β1γδ and α3β4 nAChRs (IC50 ≥ 60 μM). PNU-282987 is inactive against a panel of 32 receptors at 1 μM, except 5-HT3 receptors (Ki = 930 nM).
Pathways	Ion Channel/Membrane Transporter Neuro Signaling Pathway
Targets	nAChR

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