沙格列汀盐酸盐
| CAS号 | 709031-78-7 | 货号 | BCP21271 |
| 中文名 | 沙格列汀盐酸盐 | ||
| 英文名 | Saxagliptin hydrochloride | ||
| 中文别名 | 盐酸沙格列汀; | ||
| 英文别名 | Saxagliptin HCl;BMS477118; BMS 477118; BMS-477118; | ||
| 分子式 | C18H26ClN3O2 | 分子量 | 351.87 |
| 生物活性 | Saxagliptin Hydrochloride is the hydrochloride salt form of saxagliptin, an orally bioavailable, potent, selective and competitive, cyanopyrrolidine-based inhibitor of dipeptidyl peptidase 4 (DPP-4), with hypoglycemic activity. Saxagliptin is metabolized into an, although less potent, active mono-hydroxy metabolite.Saxagliptin is a new oral hypoglycemic (anti-diabetic drug) of the new dipeptidyl peptidase-4 (DPP-4) inhibitor class of drugs. Saxagliptin was approved in 2008 for the treatment of type 2 diabetes. Saxagliptin is a competitive DPP4 inhibitor that slows the inactivation of the incretin hormones, thereby increasing their bloodstream concentrations and reducing fasting and postprandial glucose concentrations in a glucose-dependent manner in patients with type 2 diabetes mellitus. . | ||
| 信号通路 | Protease/Metabolic Enzyme | ||
| 靶 点 | DPP | ||
结构式
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