SB 243213

  • Chemical Properties
CAS No. 200940-22-3 Cat. No. BCP43353
Name SB 243213
Synonyms SB-243213; SB243213;
Formula C22H19F3N4O2 M. Wt 428.41
  • Biological Activity
Description SB 243213 is an orally active, selective and high-affinity 5-HT2C receptor antagonist with a pKi of 9.37 and a pKb of 9.8 for human 5-HT2C receptor. SB 243213 shows greater than a 100-fold selectivity over a wide range of neurotransmitter receptors, enzymes and ion channels. SB 243213 has improved anxiolytic profile and has the potential for schizophrenia and motor disorders.
Pathways GPCR/G Protein 
Targets 5 HT Receptor/Serotonin Receptor 

Structure

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