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Nature products
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Intermediate
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Raw Materials
5 HT Receptor/Serotonin Receptor
Chemical Structure | Cat. No. | Product Name | CAS No. |
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BCP24269 | Temanogrel New | 887936-68-7 |
Temanogrel is a highly selective 5-HT2A receptor antagonist with a Ki of 4.9 nM.
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BCP49052 | NAS-181 methanesulfonate New | 205242-62-2 |
NAS-181 methanesulfonate is a 5-HT(1B) receptor antagonist.
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BCP24751 | Sarizotan New | 351862-32-3 |
Sarizotan is an orally active serotonin 5-HT1A receptor and dopamine receptor agonist. Sarizotan (EMD 128130) exhibits IC50 values of 6.5 nM (rat 5-HT1A), 0.1 nM (human 5-HT1A), 15.1 nM (rat D2), 17 nM (human D2), 6.8 nM (human D3) and 2.4 nM (human D4.2), respectively.
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BCP48961 | Opiranserin New | 1441000-45-8 |
Opiranserin is a glycine transporter inhibitor and serotonin receptor antagonist. Opiranserin is a drug candidate.
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BCP25643 | DOI hydrochloride New | 42203-78-1 |
DOI hydrochloride is a brain penetrant, mixed 5-HT2A/5-HT2C receptor agonist (Ki values are 0.7, 2.4 and 20 nM for 5-HT2A, 5-HT2C and 5-HT2B receptors respectively). Reduces rapid eye movement (REM) and slow wave sleep and increases waking in the rat. Hallucinogenic agent. Acts via 5-HT2A receptors to inhibit the inflammatory effects of tumor necrosis factor (TNF)-α.
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BCP25681 | 8-OH-Dpat New | 78950-78-4 |
8-OH-DPAT is a potent and selective 5-HT agonist, with a pIC50 of 8.19 for 5-HT1A and a Ki of 466 nM for 5-HT7; 8-OH-DPAT weakly binds to 5-HT1B (pIC50, 5.42), 5-HT (pIC50 <5).
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BCP48408 | Prucalopride hydrochloride New | 179474-80-7 |
Prucalopride hydrochloride is a selective 5-HT4 agonist.
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BCP48648 | RU-24969 New | 66611-26-5 |
RU-24969 is a potent, selective agonist of 5-HT1A and 5-HT1B receptors, with preference for 5-HT1B.
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BCP48214 | (Z)-Thiothixene New | 3313-26-6 |
Thiothixene is a modulator of human P-glycoprotein and is frequently used a an anti-psychotic.
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BCP48258 | WAY-161503 New | 75704-24-4 |
WAY-161503 is a full agonist of 5-HT2C receptors that exhiits ~6-fold less potent at 5-HT2A receptors (Ki = 18 nM) and 20-fold less potent at 5-HT2B receptors (Ki = 60 nM).
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