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Nature products
Antibodies
Peptides
Catalysts
Impurities
Intermediate
- Amino acid
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Raw Materials
CGRP Receptor
Chemical Structure | Cat. No. | Product Name | CAS No. |
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BCP42168 | Rimegepant sulfate hydrate New | 1374024-48-2 |
Rimegepant is a potent, selective, competitive, and orally active calcitonin gene-related peptide (CGRP) antagonist in clinical trials for treating migraines.
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BCP29403 | BIBN 4096BS | 204697-65-4 |
BIBN 4096BS is the first potent and selective non-peptide antagonist of the calcitonin gene-related peptide 1 (CGRP1) receptor with IC50 of 0.03 nM and with a Ki of 14.4 pM for human CGRP.
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BCP28575 | BMS 927711 New | 1289023-67-1 |
Rimegepant is a highly potent, oral calcitonin gene-related peptide (CGRP) receptor antagonist with a Ki value of 0.027 nM.
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BCP29018 | MK-8031 | 1374248-81-3 |
MK-8031, also known as Atogepant, is a calcitonin gene-related peptide receptor antagonist.
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BCP27622 | MK-3207 HCl | 957116-20-0 |
MK-3207 (Hydrochloride) is a potent and orally bioavailable CGRP receptor antagonist with IC50 of 0.12 nM and Ki of 0.024 nM, and is highly selective versus human AM1, AM2, CTR, and AMY3.
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BCP07257 | Telcagepant | 781649-09-0 |
MK-0974 is a highly potent, selective, and orally bioavailable CGRP receptor antagonist, which may be valuable in the acute treatment of migraine.
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BCP02225 | MK 3207 | 957118-49-9 |
MK-3207 is a potent and orally bioavailable CGRP receptor antagonist. In common with other CGRP receptor antagonists, MK-3207 displays lower affinity for human CGRP receptors from other species, including canine and rodent.
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