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Histone Methyltransferase

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Histone Methyltransferase

Chemical Structure Cat. No. Product Name CAS No.
BAY-598 R-isomer Chemical Structure
BCP44956 BAY-598 R-isomer 1906920-28-2
BAY-598 R-isomer is the R-isomer of BAY589.
SGC3027 Chemical Structure
BCP44921 SGC3027 2624313-13-7
SGC3027 is a histone methyltransferase inhibitor.
MRTX-1719 Chemical Structure
BCP44551 MRTX-1719 2630904-45-7
MRTX1719 is a first-in-class MTA-cooperative PRMT5 inhibitor that selectively elicits antitumor activity in MTAP/CDKN2A deleted cancer models
Dot1L-IN-4 Chemical Structure
BCP43459 Dot1L-IN-4 2565705-02-2
Dot1L-IN-4 is a potent disruptor of telomeric silencing 1-like protein (DOT1L) inhibitor.
BRD0639 Chemical Structure
BCP43480 BRD0639 BRD0639
BRD0639 is a potent PRMT5 inhibitor.
TP-064 Chemical Structure
BCP43164 TP-064 2080306-20-1
TP-064 is a potent, selective, and cell-active inhibitor of PRMT4 with IC50 of <10 nM and Kd of 7.1 nM, shows high selectivity (>100-fold) for PRMT4 over other PRMTs.
MRK-740 Chemical Structure
BCP40609 MRK-740 2387510-80-5
MRK-740 is a potent, selective and substrate-competitive PRDM9 histone methyltransferase inhibitor.
LLY-283 Chemical Structure
BCP39701 LLY-283 2040291-27-6
LLY-283 is an inhibitor of protein arginine methyltransferase 5 (PRMT5) with antitumor activity. It potently suppresses cancer growth via inhibiting PRMT5 expressed in breast cancer, gastric cancer, glioblastoma, and lymphoma cells.
Tazemetostat hydrobromide Chemical Structure
BCP39175 Tazemetostat hydrobromide 1467052-75-0
Tazemetostat is a potent, selective, and orally bioavailable small-molecule inhibitor of EZH2 enzymatic activity.
BIX 01294 trihydrochloride hydrate Chemical Structure
BCP38667 BIX 01294 trihydrochloride hydrate 1808255-64-2
BIX 01294 trihydrochloride hydrate, a diazepin-quinazolinamine derivative, is a histone-lysine methyltransferase (HMTase) inhibitor that modulates the epigenetic status of chromatin.
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