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GPCR/G Protein
Endothelin Receptor

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Endothelin Receptor

Chemical Structure Cat. No. Product Name CAS No.
Sparsentan Chemical Structure
BCP23969 Sparsentan 254740-64-2
Sparsentan is a highly potent dual angiotensin II and endothelin A receptor antagonist with Kis of 0.8 and 9.3 nM, respectively.
TAK 044 Chemical Structure
BCP37381 TAK 044 157380-72-8
TAK-044 has been found to be an endothelin receptor antagonist that was once studied against some sort of liver disorders and subarachnoid haemorrhage.
BMS-182874 Hydrochloride Chemical Structure
BCP33050 BMS-182874 Hydrochloride 1215703-04-0
BMS 182874 hydrochloride is a potent, selective and competitive non-peptide endothelin ETA receptor antagonist (Ki = 48 nM).
BQ-788 Chemical Structure
BCP29520 BQ-788 173326-37-9
BQ788 is a endothelin B receptor antagonist. BQ788 attenuates stab wound injury-induced reactive astrocytes in rat brain. BQ788 were well tolerated and showed signs of directly and indirectly reducing the viability of melanoma cells.
Carperitide Chemical Structure
BCP12639 Carperitide 89213-87-6
Carperitide is a polypeptide.
Darusentan Chemical Structure
BCP13024 Darusentan 171714-84-4
Darusentan (LU-135252; HMR-4005) is an endothelin receptor antagonist.
Hydroxy Bosentan Chemical Structure
BCP15832 Hydroxy Bosentan 253688-60-7
Hydroxy Bosentan is a metabolite of Bosentan.
Aprocitentan Chemical Structure
BCP28125 Aprocitentan 1103522-45-7
Aprocitentan is the major and pharmacologically active metabolite of macitentan, which is dual ETA/ETB antagonist designed for tissue targeting.
BQ-123 Chemical Structure
BCP29354 BQ-123 136553-81-6
BQ-123 is a elective ETA endothelin receptor antagonist (Ki values are 1.4 and 1500 nM at ETA and ETB receptors respectively).
Ro 46-2005 Chemical Structure
BCP17756 Ro 46-2005 150725-87-4
Ro 46-2005 is a novel synthetic non-peptide endothelin receptor antagonist, inhibits the specific binding of 125I-ET-1 to human vascular smooth muscle cells (ETA receptor) with IC50 of 220 nM.
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