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GPCR/G Protein

Chemical Structure Cat. No. Product Name CAS No.
CJ033466 Chemical Structure
 BCP46275 CJ033466 519148-48-2
CJ-033466 is a Serotonin 5-HT4 Receptor Agonist.
GLUT inhibitor-1 Chemical Structure
 BCP46268 GLUT inhibitor-1 2421141-40-2
GLUT inhibitor-1 is a potent and orally active inhibitor of glucose transporters, targeting both GLUT1 and GLUT3 , with IC 50 s of 242 nM and 179 nM, respectively.
Chemical Structure
Retosiban Chemical Structure
 BCP46037 Retosiban 820957-38-8
Retosiban is an oral drug which acts as a selective, sub-nanomolar (Ki = 0.65 nM) oxytocin receptor antagonist with >1400-fold selectivity over the related vasopressin receptors.
Sigma-1 receptor antagonist 2 Chemical Structure
 BCP46031 Sigma-1 receptor antagonist 2 1639220-15-7
Sigma-1 receptor antagonist 2 is a potent and selective sigma 1 receptor (σ1 R) antagonist with Kis of 3.88 and 1288 nM for σ1 and σ2 receptor, respectively.
MRTX0902 Chemical Structure
 BCP46021 MRTX0902 2654743-22-1
MRTX0902 is an effective SOS1 inhibitor with an IC50 of 46 nM.
CS-003 Chemical Structure
 BCP45999 CS-003 191672-52-3
CS-003 is a triple tachykinin receptor antagonist, shows high affinities for human (Neurokinin) NK1, NK2 and NK3 receptors with Ki values of 2.3 nM, 0.54 nM and 0.74 nM, respectively.
Ro60-0175 Chemical Structure
 BCP45982 Ro60-0175 169675-08-5
Ro60-0175 is a potent and selective agonist of 5-HT2C receptor.
BAY 60-6583 Chemical Structure
 BCP45903 BAY 60-6583 910487-58-0
BAY 60-6583 is a potent and high-affinity agonist of adenosine A2B receptor (EC50 = 3 nM) over A1, A2A, and A3 receptors. BAY 60-6583 binds to mouse, rabbit, and dog A2BAR with Ki values of 750 nM, 340 nM and 330 nM, respectively. BAY 60-6583 has a cardioprotective effect in a myocardial ischemia model.
PF-4479745 Chemical Structure
 BCP45867 PF-4479745 1065110-43-1
PF-4479745 is a potent and selective 5-HT2C agonist (EC50 = 10 nM).
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