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PI3K

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PI3K

Chemical Structure Cat. No. Product Name CAS No.
Gilmelisib Chemical Structure
 BCP46378 Gilmelisib 1845777-61-8
Gilmelisib is a PI3K inhibitor and antineoplastic.
GSK251 Chemical Structure
 BCP46226 GSK251 2125968-05-8
GSK251 is a highly potent, highly selective, orally bioavailable inhibitor of PI3Kδ with a novel binding mode.
ETP-45658 Chemical Structure
 BCP45165 ETP-45658 1198357-79-7
ETP-45658 is a PI3-kinase inhibitor, also ihibiting DNA-PK and mTOR.
GS-9901 Chemical Structure
 BCP44115 GS-9901 1640247-87-5
GS-9901 is a potent, orally active and highly selective inhibitor of PI3Kδ (PI3Kdelta IC50 = 1.0nM, HWB delta EC50 = 1.5 nM; CLpr hHep = 0.05 L/h/kg.).
Panulisib Chemical Structure
 BCP44105 Panulisib 1356033-60-7
Panulisib is an orally bioavailable inhibitor of phosphoinositide 3-kinase (PI3K), mammalian target of rapamycin (mTOR), activin receptor-like kinase 1 (ALK-1) and DNA-dependent protein kinase (DNA-PK), with potential anti-angiogenic and antineoplastic activities.
Parsaclisib hydrochloride Chemical Structure
 BCP42656 Parsaclisib hydrochloride 1995889-48-9
Parsaclisib, also known as INCB050465, is a novel PI3Kδ inhibitor which synergizes with PIM protein kinase inhibition to cause tumor regression in a model of DLBCL.
PIK-108 Chemical Structure
 BCP41853 PIK-108 901398-68-3
PIK-108 is an allosteric inhibitor of the lipid modifying kinases, phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunits β and δ (PI3Kβ/δ).
SRX3207 Chemical Structure
 BCP40266 SRX3207 2254693-15-5
SRX3207 is an orally active dual inhibitor of Syk-PI3K with IC50 of 39.9 nM, 31200 nM, 3070 nM, 3070 nM, 244 nM, 388 nM, 9790 nM for Syk, Zap70, BRD41, BRD42, PI3K alpha, PI3K delta, PI3K gamma, respectively.
IPI-3063 Chemical Structure
 BCP39855 IPI-3063 1425043-73-7
IPI-3063 is a potent and selective phosphoinoside-3-kinase (PI3K) p110δ inhibitor. IPI-3063 was shown to inhibit mouse B cell proliferation, survival, and plasmablast differentiation, and also inhibit human B cell proliferation in vitro.
Nemiralisib Chemical Structure
 BCP38658 Nemiralisib 1254036-71-9
Nemiralisib, also known as GSK2269557, is a highly potent and selective inhaled PI3Kδ inhibitor for the treatment of COPD.
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