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Signaling Pathways
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Protease/Metabolic Enzyme
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Research Areas
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Nature products
Antibodies
Peptides
Catalysts
Impurities
Intermediate
- Amino acid
- Ammonia Series
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- Azaindazole
- Nucleoside Series
- Quinazoline
- Pyrazole Series
- Quinoline Series
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- Boric acid
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- Thiophene Series
- Saccharide
- Azaindole
- Indole Series
- Indazole Series
- Piperidine Series
- Heterocyclic Series
- Pyridine Series
- Benzene Series
Raw Materials
Histamine Receptor
Chemical Structure | Cat. No. | Product Name | CAS No. |
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BCP44465 | Antazoline phosphate New | 154-68-7 |
Antazoline phosphate is an antihistamine with anticholinergic properties used to relieve nasal congestion and the symptoms of allergic conjunctivitis. Antazoline is an ethylenediamine derivative with histamine H1 antagonistic and sedative properties. Antazoline antagonizes histamine H1 receptor and prevents the typical allergic symptoms caused by histamine activities on capillaries, skin, mucous membranes, and gastrointestinal and bronchial smooth muscles.
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BCP43974 | Terfenadine New | 50679-08-8 |
Terfenadine is a potent open-channel blocker of hERG with a mean IC50 of 204 nM.
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BCP43719 | Pimethixene New | 314-03-4 |
Pimethixene is antihistamine and anticholinergic of the thioxanthene chemical class that is often used to treat hyperactivity, anxiety, sleep disorders, and allergy. It is also used for anesthesia and as a bronchodilator (to dilate the bronchi and bronchioles for more airflow).
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BCP43718 | Pimethixene maleate New | 13187-06-9 |
Pimethixene maleate is antihistamine and antiserotonergic compound, acts as an antimigraine agent. Pimethixene maleate is a highly potent antagonist of 5-HT1A, 5-HT2A, 5-HT2B, 5-HT2C, histamine H1, dopamine D2 and D4.4 as well as muscarinic M1 and M2 receptors, with pKis of 7.63, 10.22, 10.44, 8.42, 10.14, 8.19, 7.54, 8.61 and 9.38, respectively.
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BCP43687 | Chlorphenoxamine New | 77-38-3 |
Chlorphenoxamine is a diarylmethane. It has a role as an anticoronaviral agent.
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BCP39480 | Thioperamide New | 106243-16-7 |
Thioperamide is a potent histamine H3 and H4 antagonist/inverse agonist (Ki = 25 and 27 nM for human recombinant H3 and H4 receptors, respectively). Thioperamide can cross the blood-brain barrier freely.
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BCP39479 | Thioperamide maleate New | 148440-81-7 |
Thioperamide maleate is a selective histamine H3 receptor antagonist that crosses the blood-brain barrier.
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BCP37369 | JNJ-5207852 New | 398473-34-2 |
JNJ-5207852 is a selective and potent histamine H3 receptor (H3R) antagonist, with pKis of 8.9, 9.24 for rat and human H3R, respectively.
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BCP25799 | Thonzylamine New | 91-85-0 |
Thonzylamine is a first-generation ethylenediamine H1-antihistamine.
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BCP33258 | Doxepin-d3 Hydrochloride New | 347840-07-7 |
Doxepin D3 Hydrochloride is a deuterium labeled Doxepin Hydrochloride.Doxepin is a tricyclic antidepressant (TCA) used for the treatment of major depression and anxiety.
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