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Histamine Receptor

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Histamine Receptor

Chemical Structure Cat. No. Product Name CAS No.
Antazoline phosphate Chemical Structure
 BCP44465 Antazoline phosphate 154-68-7
Antazoline phosphate is an antihistamine with anticholinergic properties used to relieve nasal congestion and the symptoms of allergic conjunctivitis. Antazoline is an ethylenediamine derivative with histamine H1 antagonistic and sedative properties. Antazoline antagonizes histamine H1 receptor and prevents the typical allergic symptoms caused by histamine activities on capillaries, skin, mucous membranes, and gastrointestinal and bronchial smooth muscles.
Terfenadine Chemical Structure
 BCP43974 Terfenadine 50679-08-8
Terfenadine is a potent open-channel blocker of hERG with a mean IC50 of 204 nM.
Pimethixene Chemical Structure
 BCP43719 Pimethixene 314-03-4
Pimethixene is antihistamine and anticholinergic of the thioxanthene chemical class that is often used to treat hyperactivity, anxiety, sleep disorders, and allergy. It is also used for anesthesia and as a bronchodilator (to dilate the bronchi and bronchioles for more airflow).
Pimethixene maleate Chemical Structure
 BCP43718 Pimethixene maleate 13187-06-9
Pimethixene maleate is antihistamine and antiserotonergic compound, acts as an antimigraine agent. Pimethixene maleate is a highly potent antagonist of 5-HT1A, 5-HT2A, 5-HT2B, 5-HT2C, histamine H1, dopamine D2 and D4.4 as well as muscarinic M1 and M2 receptors, with pKis of 7.63, 10.22, 10.44, 8.42, 10.14, 8.19, 7.54, 8.61 and 9.38, respectively.
Chlorphenoxamine Chemical Structure
 BCP43687 Chlorphenoxamine 77-38-3
Chlorphenoxamine is a diarylmethane. It has a role as an anticoronaviral agent.
Thioperamide Chemical Structure
 BCP39480 Thioperamide 106243-16-7
Thioperamide is a potent histamine H3 and H4 antagonist/inverse agonist (Ki = 25 and 27 nM for human recombinant H3 and H4 receptors, respectively). Thioperamide can cross the blood-brain barrier freely.
Thioperamide maleate Chemical Structure
 BCP39479 Thioperamide maleate 148440-81-7
Thioperamide maleate is a selective histamine H3 receptor antagonist that crosses the blood-brain barrier.
JNJ-5207852 Chemical Structure
 BCP37369 JNJ-5207852 398473-34-2
JNJ-5207852 is a selective and potent histamine H3 receptor (H3R) antagonist, with pKis of 8.9, 9.24 for rat and human H3R, respectively.
Thonzylamine Chemical Structure
 BCP25799 Thonzylamine 91-85-0
Thonzylamine is a first-generation ethylenediamine H1-antihistamine.
Doxepin-d3 Hydrochloride Chemical Structure
 BCP33258 Doxepin-d3 Hydrochloride 347840-07-7
Doxepin D3 Hydrochloride is a deuterium labeled Doxepin Hydrochloride.Doxepin is a tricyclic antidepressant (TCA) used for the treatment of major depression and anxiety.
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