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Hormone Pathay

Chemical Structure Cat. No. Product Name CAS No.
ARD2585 Chemical Structure
 BCP46972 ARD2585 ARD2585
ARD-2585 is an exceptionally potent and orally active PROTAC degrader of androgen receptor.
NH-3 Chemical Structure
 BCP46931 NH-3 447415-26-1
NH-3 is an orally active, reversible thyroid hormone receptor (THR) antagonist with an IC50 of 55 nM.
2-Hydroxyestrone Chemical Structure
 BCP46743 2-Hydroxyestrone 362-06-1
2-Hydroxyestrone, a specific receptor-mediated antiestrogenic agent with anticarcinogenic activity, inhibits the proliferation of estrogen receptor-positive MCF-7, but not estrogen receptor-negative MDA-MB-231.
BMS-986122 Chemical Structure
 BCP46445 BMS-986122 313669-88-4
BMS-986122 is a positive allosteric modulator of the μ-Opioid Receptor.
ARV-471 Chemical Structure
 BCP45881 ARV-471 2229711-08-2
ARV-471 is a best-in-class, orally active estrogen receptor (ER) PROTAC degrader.
ML 145 Chemical Structure
 BCP45167 ML 145 1164500-72-4
ML 145 is a selective antagonist for the GPR35 orphan receptor GPCR (IC50 = 20.1 nM). Over 1000-fold more selective for GPR35 compared to GPR55 antagonists.
Difelikefalin TFA Chemical Structure
 BCP44865 Difelikefalin TFA 2742623-88-5
Difelikefalin is a κ-opioid receptor (KOR) agonist. It activates KOR in HEK293 cells expressing the human receptor (EC50 = 0.16 nM in a transactivation assay) and inhibits forskolin-induced cAMP production in R1.G1 mouse thyoma cells (EC50 = 0.048 nM).
Amcenestrant Chemical Structure
 BCP38455 Amcenestrant 2114339-57-8
Amcenestrant (SAR439859) is an orally available and nonsteroidal selective estrogen receptor degrader (SERD) with potential antineoplastic activity. SAR439859 is a potent estrogen receptor (ER) antagonist with EC50 of 0.2 nM for ERα degradation.
U-54494A Chemical Structure
 BCP44497 U-54494A 92953-41-8
U-54494A is a κ-opioid agonist and a potential NMDA antagonist. U-54494A hydrochloride is used as an anticonvulsant.
Difelikefalin HCl Chemical Structure
 BCP44189 Difelikefalin HCl 2413256-25-2
Difelikefalin is a novel and potent kappa opioid receptor agonist.
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