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Epigenetic Reader Domain

Chemical Structure Cat. No. Product Name CAS No.
EML 425 Chemical Structure
 BCP46797 EML 425 1675821-32-5
EML425 is a potent and selective CREB binding protein (CBP)/p300 inhibitor with IC50s of 2.9 and 1.1 μM, respectively.
CFT-8634 Chemical Structure
 BCP46564 CFT-8634 2704617-96-7
CFT-8634 is a degrader targeting BRD9 extracted from patent WO2021178920A1 compound 173.
GSK1379725A Chemical Structure
 BCP46513 GSK1379725A 1802251-00-8
GSK1379725A is the first selective inhibitor of BPTF over Brd4.
BAZ1A-IN-1 Chemical Structure
 BCP46449 BAZ1A-IN-1 941521-45-5
BAZ1A-IN-1 is a potent inhibitor of BAZ1A (bromodomain-containing protein). BAZ1A-IN-1 shows a KD value of 0.52 μM against BAZ1A bromodomain.
M-525 Chemical Structure
 BCP46311 M-525 2173582-08-4
M-525 is a first-in-class, highly potent, irreversible small-molecule inhibitor of the menin-MLL interaction.
dBRD9 Chemical Structure
 BCP45901 dBRD9 2170679-45-3
dBRD9 is a potent and selective BRD9 bromodomain degrader composed of the BRD9 inhibitor BI 7273 conjugated to the cereblon E3 ligase ligand pomalidomide.
I-BET567 Chemical Structure
 BCP45484 I-BET567 1887237-54-8
I-BET567 is a potent and orally active inhibitor of pan-BET candidate with pIC50s of 6.9 and 7.2 for BRD4 BD1 and BD2, respectively.
Bet-IN-4 Chemical Structure
 BCP45446 Bet-IN-4 1801503-93-4
Bet-IN-4 is a highly potent, selective and orally active pan-BET inhibitor that has shown preclinical evidence of tumour growth inhibition in breast cancer and in leukaemia and prostate cancer xenograft models.
CTB Chemical Structure
 BCP45206 CTB 451491-47-7
CTB (Cholera Toxin B subunit) is an activator of p300 histone acetyltransferase and induces apoptosis in MCF-7 cells.
PROTAC BRD4 ligand-1 Chemical Structure
 BCP45084 PROTAC BRD4 ligand-1 2313230-51-0
PROTAC BRD4 ligand-1 is a potent inhibitor of BET .
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