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Epigenetic Reader Domain

Chemical Structure Cat. No. Product Name CAS No.
BMS 986158 Chemical Structure
 BCP25147 BMS 986158 1800340-40-2
BMS-986158 is an inhibitor of the bromodomain and extra-terminal (BET) proteins.
SRX3177 Chemical Structure
 BCP48567 SRX3177 2241237-51-2
SRX3177 is a novel potent triple action inhibitor, targeting BRD, PI3K, and CDK.
AU-15330 Chemical Structure
 BCP46987 AU-15330 2380274-50-8
AU-15330 is a novel, highly specific and VHL-dependent PROTAC degrader of SWI/SNF ATPase components (SMARCA2, SMARCA4 and PBRM1) that shows preferential cytotoxicity in enhancer-binding transcription factor-addicted cancers at low nanomolar concentrations.
EML 425 Chemical Structure
 BCP46797 EML 425 1675821-32-5
EML425 is a potent and selective CREB binding protein (CBP)/p300 inhibitor with IC50s of 2.9 and 1.1 μM, respectively.
CFT-8634 Chemical Structure
 BCP46564 CFT-8634 2704617-96-7
CFT-8634 is a degrader targeting BRD9 extracted from patent WO2021178920A1 compound 173.
GSK1379725A Chemical Structure
 BCP46513 GSK1379725A 1802251-00-8
GSK1379725A is the first selective inhibitor of BPTF over Brd4.
BAZ1A-IN-1 Chemical Structure
 BCP46449 BAZ1A-IN-1 941521-45-5
BAZ1A-IN-1 is a potent inhibitor of BAZ1A (bromodomain-containing protein). BAZ1A-IN-1 shows a KD value of 0.52 μM against BAZ1A bromodomain.
M-525 Chemical Structure
 BCP46311 M-525 2173582-08-4
M-525 is a first-in-class, highly potent, irreversible small-molecule inhibitor of the menin-MLL interaction.
dBRD9 Chemical Structure
 BCP45901 dBRD9 2170679-45-3
dBRD9 is a potent and selective BRD9 bromodomain degrader composed of the BRD9 inhibitor BI 7273 conjugated to the cereblon E3 ligase ligand pomalidomide.
I-BET567 Chemical Structure
 BCP45484 I-BET567 1887237-54-8
I-BET567 is a potent and orally active inhibitor of pan-BET candidate with pIC50s of 6.9 and 7.2 for BRD4 BD1 and BD2, respectively.
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