Home   >  
Ion Channel/Membrane Transporter
  >  
MCT

Classified by application

All Products

Signaling Pathways

Research Areas

Nature products

Antibodies

Peptides

Catalysts

Impurities

Intermediate

Raw Materials

MCT

Chemical Structure Cat. No. Product Name CAS No.
AZD0095 Chemical Structure
BCP49600 AZD0095 2750001-23-9
AZD0095 is a selective and orally active MCT4 inhibitor (IC50: 1.3 nM).
AR-C117977 Chemical Structure
BCP23781 AR-C117977 216685-07-3
AR-C117977 is a potent MCT1 inhibitor, which can reduce vimmune responses both in vitro and in vivo, maintains long-term graft survival, and induces operational tolerance.
VB-124 Chemical Structure
BCP48843 VB-124 2230186-18-0
VB124 is a novel, highly potent MCT4 inhibitor that mitigated hypertrophy in cultured cardiomyocytes and in mice.
AZD3965 Chemical Structure
BCP09948 AZD3965 733809-45-5
AZD3965 is a selective inhibitor of monocarboxylate transporter 1 (MCT1) with a binding affinity of 1.6 nM, is 6 fold selective over MCT2 and does not inhibit MCT4 at 10 μM.
AZD3965 Chemical Structure
BCP17734 AZD3965 1448671-31-5
AZD3965 is a selective inhibitor of monocarboxylate transporter 1 (MCT1) with a binding affinity of 1.6 nM, is 6 fold selective over MCT2 and does not inhibit MCT4 at 10 μM.
AR-C155858 Chemical Structure
BCP13211 AR-C155858 496791-37-8
AR-C155858 is a novel inhibitor of the monocarboxylate transporters (MCTs) MCT1 and MCT2 (Ki values are 2.3 and <10 nM respectively); exhibits no activity at MCT4.
7ACC2 Chemical Structure
BCP11646 7ACC2 1472624-85-3
7ACC2 is a new potent MCT inhibitor with IC50 of 11 nM for inhibition of [14C]-lactate influx; new antitumor treatment targeting lactate transport in cancer cells.
BAY-8002 Chemical Structure
BCP30742 BAY-8002 724440-27-1
BAY-8002 is a potent, selective, orally active inhibitor of monocarboxylate transporter 1 (MCT1), with an IC50 of 85 nM in the MCT1-expressing DLD-1 cells, displays excellent selectivity against MCT4. Anti-tumor activity.
0086-13720134139