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Opioid Receptor

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Opioid Receptor

Chemical Structure Cat. No. Product Name CAS No.
CTOPA Chemical Structure
 BCP24191 CTOPA 103429-31-8
CTOP is a potent and selective μ opioid receptor antagonist (Ki values are 0.96 and >10,000 nM for μ and δ receptors respectively).
Bevenopran Chemical Structure
 BCP48962 Bevenopran 676500-67-7
Bevenopran is a peripheral μ-opioid receptor antagonist.
Axelopran Chemical Structure
 BCP47463 Axelopran 949904-48-7
Axelopran, also known as TD-1211, is a potent, selective, and peripherally-restricted μ-, κ-, and δ-opioid receptor antagonist, with similar affinity for the μ- and κ-opioid receptors and about an order of magnitude lower affinity for the δ-opioid recept
BMS-986122 Chemical Structure
 BCP46445 BMS-986122 313669-88-4
BMS-986122 is a positive allosteric modulator of the μ-Opioid Receptor.
Difelikefalin TFA Chemical Structure
 BCP44865 Difelikefalin TFA 2742623-88-5
Difelikefalin is a κ-opioid receptor (KOR) agonist. It activates KOR in HEK293 cells expressing the human receptor (EC50 = 0.16 nM in a transactivation assay) and inhibits forskolin-induced cAMP production in R1.G1 mouse thyoma cells (EC50 = 0.048 nM).
U-54494A Chemical Structure
 BCP44497 U-54494A 92953-41-8
U-54494A is a κ-opioid agonist and a potential NMDA antagonist. U-54494A hydrochloride is used as an anticonvulsant.
Difelikefalin HCl Chemical Structure
 BCP44189 Difelikefalin HCl 2413256-25-2
Difelikefalin is a novel and potent kappa opioid receptor agonist.
DAMGO Chemical Structure
 BCP42954 DAMGO 78123-71-4
DAMGO is a μ-opioid receptor (μ-OPR ) selective agonist with a Kd of 3.46 nM for native μ-OPR.
Difelikefalin acetate Chemical Structure
 BCP42797 Difelikefalin acetate 1024829-44-4
Difelikefalin is an intravenous agent for the treatment of postoperative pain.
Difelikefalin Chemical Structure
 BCP24752 Difelikefalin 1024828-77-0
Difelikefalin is a peripherally restricted and selective agonist of kappa opioid receptor (KOR). Difelikefalin produces anti-inflammatory effects and has the potential in modulating pruritus in conditions such as chronic kidney disease.
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