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Opioid Receptor

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Opioid Receptor

Chemical Structure Cat. No. Product Name CAS No.
Naloxone HCl Chemical Structure
 BCP06880 Naloxone HCl 357-08-4
Naloxone hydrochloride is a hydrochloride resulting from the formal reaction of equimolar amounts of naloxone and hydrogen chloride. A specific opioid antagonist, it is used to reverse the effects of opioids, both following their use of opioids during surgery and in cases of known or suspected opioid overdose. It has a role as an antidote to opioid poisoning, a mu-opioid receptor antagonist and a central nervous system depressant. It contains a naloxone(1+).
CTOPA Chemical Structure
 BCP24191 CTOPA 103429-31-8
CTOP is a potent and selective μ opioid receptor antagonist (Ki values are 0.96 and >10,000 nM for μ and δ receptors respectively).
Bevenopran Chemical Structure
 BCP48962 Bevenopran 676500-67-7
Bevenopran is a peripheral μ-opioid receptor antagonist.
Axelopran Chemical Structure
 BCP47463 Axelopran 949904-48-7
Axelopran, also known as TD-1211, is a potent, selective, and peripherally-restricted μ-, κ-, and δ-opioid receptor antagonist, with similar affinity for the μ- and κ-opioid receptors and about an order of magnitude lower affinity for the δ-opioid recept
BMS-986122 Chemical Structure
 BCP46445 BMS-986122 313669-88-4
BMS-986122 is a positive allosteric modulator of the μ-Opioid Receptor.
Difelikefalin TFA Chemical Structure
 BCP44865 Difelikefalin TFA 2742623-88-5
Difelikefalin is a κ-opioid receptor (KOR) agonist. It activates KOR in HEK293 cells expressing the human receptor (EC50 = 0.16 nM in a transactivation assay) and inhibits forskolin-induced cAMP production in R1.G1 mouse thyoma cells (EC50 = 0.048 nM).
U-54494A Chemical Structure
 BCP44497 U-54494A 92953-41-8
U-54494A is a κ-opioid agonist and a potential NMDA antagonist. U-54494A hydrochloride is used as an anticonvulsant.
Difelikefalin HCl Chemical Structure
 BCP44189 Difelikefalin HCl 2413256-25-2
Difelikefalin is a novel and potent kappa opioid receptor agonist.
DAMGO Chemical Structure
 BCP42954 DAMGO 78123-71-4
DAMGO is a μ-opioid receptor (μ-OPR ) selective agonist with a Kd of 3.46 nM for native μ-OPR.
Difelikefalin acetate Chemical Structure
 BCP42797 Difelikefalin acetate 1024829-44-4
Difelikefalin is an intravenous agent for the treatment of postoperative pain.
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