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GPCR/G Protein

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Chemical Structure Cat. No. Product Name CAS No.
SB-756050 Chemical Structure
BCP32623 SB-756050 447410-57-3
SB-756050 is a selective TGR5 agonist. SB756050 has the potential for type 2 diabetes treatment.
SBI-115 Chemical Structure
BCP32736 SBI-115 882366-16-7
SBI-115 is a TGR5 (GPCR19) antagonist. SBI-115 decreases hepatic cystogenesis with polycystic liver diseases via inhibiting TGR5.
TGR5 Receptor Agonist Chemical Structure
BCP08750 TGR5 Receptor Agonist 1197300-24-5
TGR5 Receptor Agonist, a potent TGR5(GPCR19) agonist.
BAR502 Chemical Structure
BCP19638 BAR502 1612191-86-2
BAR502 is a dual FXR and GPBAR1 agonist with IC50 values of 2 μM and 0.4 μM, respectively.
BAR501 Chemical Structure
BCP24972 BAR501 1632118-69-4
BAR501 is a potent, selective GPBAR1 (GPCR19; TGR5) agonist devoid of any FXR agonistic activity, effectively transactivates GPBAR1 in HEK293 cells with EC50 of 1 uM.
Deoxycholic acid Chemical Structure
BCP15620 Deoxycholic acid 83-44-3
Deoxycholic acid is specifically responsible for activating the G protein-coupled bile acid receptor TGR5 that stimulates brown adipose tissue (BAT) thermogenic activity.