卡普瑞林酒石酸盐新

参考资料仅供科学研究，不可用于个人用途。

货号：BCP15666CAS号：193273-69-7纯度：98%

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CAS号	193273-69-7	货号	BCP15666
中文名	卡普瑞林酒石酸盐
英文名	Capromorelin Tartrate
中文别名	酒石酸卡莫瑞林;
英文别名	CP 424391-18; CP-424,391-18; CP-424391 Tartrate;
SMILES	CC(C)(C(=O)NC(COCC1=CC=CC=C1)C(=O)N2CCC3=NN(C(=O)C3(C2)CC4=CC=CC=C4)C)N.C(C(C(=O)O)O)(C(=O)O)O
化学名称
分子式	C32H41N5O10	分子量	655.71
纯度	98%	配送	惯例下常温包邮
产品描述	Capromorelin Tartrate is an orally active, potent growth hormone secretagogue receptor (GHSR) agonist, with Ki of 7 nM for hGHS-R1a.Capromorelin, also known as CP-424,391, is a growth hormone secretagogue and ghrelin mimetic ( hGHS-R1a K(i)=7 nM, rat pituicyte EC(50)=3 nM). Initial studies have shown the drug to directly raise insulin growth factor 1 (IGF-1) and growth hormone levels. Capromorelin showed enhanced intestinal absorption in rodent models and exhibited superior pharmacokinetic properties, including high bioavailabilities in two animal species [F(rat)=65%, F(dog)=44%]. This short-duration GHS was orally active in canine models and was selected as a development candidate for the treatment of musculoskeletal frailty in elderly adults.

卡普瑞林酒石酸盐 新