所有产品分类
所有产品
信号通路
- Angiogenesis/Protein Tyrosine Kinase
- Apoptosis Pathway
- Cell Cycle/DNA Damage
- Epigenetics
-
GPCR/G Protein
- Urotensin Receptor
- Melatonin Receptor
- Neurotensin Receptor
- Motilin Receptor
- Glucose Transporter
- TGR5
- Cholecystokinin Receptor
- Adenylate Cyclase
- Oxytocin Receptor
- Somatostatin Receptor
- Bradykinin Receptor
- Melanocortin Receptor
- Guanylate Cyclase
- Imidazoline Receptor
- PAR
- Neuropeptide Receptor
- CRFR
- Sigma Receptor
- S1P Receptor
- GHSR
- PKA
- OX Receptor
- Adenosine Receptor
- Glucagon Receptor
- Prostaglandin Receptor
- GnRH Receptor
- NK Receptor
- Glucocorticoid Receptor
- Leukotriene Receptor
- P2 Receptor
- mAChR
- CGRP Receptor
- GPR
- CXCR
- Histamine Receptor
- CaSR
- Ras/Rho
- Vasopressin Receptor
- Smoothened/Smo
- mGluR
- Opioid Receptor
- Dopamine Receptor
- Cannabinoid Receptor
- Angiotensin Receptor
- Adrenergic Receptor
- SGLT
- Endothelin Receptor
- CCR
- 5 HT Receptor/Serotonin Receptor
- Hormone Pathay
- Ion Channel/Membrane Transporter
- Jak/Stat Pathway
- MAPK Pathway
- Microbiology/Virology
-
Neuro Signaling Pathway
- Imidazoline Receptor
- Monoamine Oxidase
- COMT
- Amyloid β
- NK Receptor
- Beta secretase
- AChE
- SSRI
- CaMK
- P glycoprotein
- Opioid Receptor
- Dopamine Receptor
- Adrenergic Receptor
- Histamine Receptor
- mGluR
- Gamma secretase
- Dopamine Transporter
- 5 HT Receptor/Serotonin Receptor
- P2 Receptor
- CGRP Receptor
- FAAH
- nAChR
- COX
- GABA Receptor
- mAChR
- NFκB
- PI3K/Akt/mTOR
-
Protease/Metabolic Enzyme
- Mitochondrial Metabolism
- Pyruvate Kinase
- SCD
- ALDH
- Serine Protease
- Neprilysin
- CETP
- FTase
- MLR
- MAGL
- Carbonic Anhydrase
- E1 E2 E3 Enzyme
- Elastase
- NOX
- PAI1
- ROR
- Glucokinase
- Aldose Reductase
- Tyrosinase
- FAS
- DGAT
- Lipoxygenase
- Nampt
- IDO
- IDH
- MMP
- Cathepsin
- Phosphatase
- Thrombin
- FXR
- RAR/RXR
- HMGCR
- FAAH
- Gamma secretase
- RAAS/ACE
- Caspase
- HIV Protease
- Aminopeptidase
- HCV Protease
- HSP
- Tryptophan Hydroxylase/TPH
- Factor Xa
- DPP
- Procollagen C Proteinase
- Integrase
- Phosphodiesterase/PDE
- Phospholipase
- LXR
- Cytochrome P450
- Proteasome
- ACC
- Xanthine Oxidase
- Carboxypeptidase
- 11β HSD
- COMT
- TGF beta/Smad
- Wnt/Stem Cell
- Others Pathway
研究领域
- Metabolic Disease
- Neurological Disease
- Endocrinology
- Diabetes
- Cardiovascular Disease
- Immunology
- Allergy
- Infection
- Inflammation
- Cancer
天然产物
抗体
多肽
催化剂
杂质对照品
医药中间体
基础原料
Estrogen Receptor
结构式 | 货号 | 产品名称 | CAS号 |
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BCP46743 | 2-羟雌甾酮 新 | 362-06-1 |
2-Hydroxyestrone, a specific receptor-mediated antiestrogenic agent with anticarcinogenic activity, inhibits the proliferation of estrogen receptor-positive MCF-7, but not estrogen receptor-negative MDA-MB-231.
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BCP45881 | ARV-471 新 | 2229711-08-2 |
ARV-471 is a best-in-class, orally active estrogen receptor (ER) PROTAC degrader.
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BCP38455 | Amcenestrant 新 | 2114339-57-8 |
Amcenestrant (SAR439859) is an orally available and nonsteroidal selective estrogen receptor degrader (SERD) with potential antineoplastic activity. SAR439859 is a potent estrogen receptor (ER) antagonist with EC50 of 0.2 nM for ERα degradation.
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BCP43932 | Giredestrant tartrate 新 | 2407529-33-1 |
Giredestrant, also known as GDC-9545 and RG6171, is a SERD.
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BCP42856 | E3 ligase Ligand 5 新 | 1055361-35-7 |
E3 ligase Ligand 5 is an estrogen-related receptor α (ERRα) antagonist with IC50s of 0.04 and 2.8 μM for ERRα and ERRγ, respectively.
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BCP41931 | PPT 新 | 263717-53-9 |
PPT, also known as Propyl pyrazole triol, is an estrogen receptor (ERalpha) agonist. PPT also exerts anti-diabetic effects in mouse models.
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BCP39883 | Giredestrant 新 | 1953133-47-5 |
Giredestrant is a SERD.
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BCP41267 | 反式-氯米芬柠檬酸盐 新 | 7599-79-3 |
trans-Clomiphene a non-steroidal estrogen receptor antagonist. It can be used for secondary hypogonadism in overweight men wishing to restore normal testicular function.
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BCP40562 | 氯米芬 新 | 911-45-5 |
Clomiphene is a triphenylethylene nonsteroidal ovulatory stimulant evaluated for antineoplastic activity against breast cancer. Clomiphene has both estrogenic and anti-estrogenic activities that compete with estrogen for binding at estrogen receptor sites in target tissues. This agent causes the release of the pituitary gonadotropins follicle stimulating hormone (FSH) and luteinizing hormone (LH), leading to ovulation.
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BCP39840 | 萘福昔定 新 | 1845-11-0 |
Nafoxidine is a member of naphthalenes, a ring assembly and a member of benzenes.
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