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Opioid Receptor

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Opioid Receptor

结构式 货号 产品名称 CAS号
DAMGO 结构式
BCP42954 DAMGO 78123-71-4
DAMGO is a μ-opioid receptor (μ-OPR ) selective agonist with a Kd of 3.46 nM for native μ-OPR.
Difelikefalin acetate 结构式
BCP42797 Difelikefalin醋酸盐 1024829-44-4
Difelikefalin is an intravenous agent for the treatment of postoperative pain.
Difelikefalin 结构式
BCP24752 Difelikefalin 1024828-77-0
Difelikefalin is a peripherally restricted and selective agonist of kappa opioid receptor (KOR). Difelikefalin produces anti-inflammatory effects and has the potential in modulating pruritus in conditions such as chronic kidney disease.
BMS986188 结构式
BCP37890 BMS986188 1776115-10-6
BMS-986188 is a novel Potent and Selective Positive Allosteric Modulator of the delta-Opioid Receptor.
BMS986187 结构式
BCP37889 BMS986187 684238-37-7
BMS-986187 is a novel Potent and Selective Positive Allosteric Modulators of the delta-Opioid Receptor.
ML335 结构式
BCP37811 ML335 1069498-96-9
ML-335 is an agonist for µ-opioid receptor (OPRM1)- d-opioid receptors (OPRD1) heterodimerization.
EST73502 HCl 结构式
BCP37164 EST73502 HCl 2307458-82-6
EST73502 is a Dual μ‑Opioid Receptor Agonist and σ1 Receptor Antagonist Clinical Candidate for the Treatment of Pain.
LY-2795050 结构式
BCP33958 LY-2795050 1346133-08-1
LY2795050 is a nobel kappa opioid receptor selective antagonist.
Aticaprant 结构式
BCP32123 Aticaprant 1174130-61-0
Aticaprant is a potent and centrally-penetrant kappa opioid receptor antagonist with a Ki of 0.807 nM.
BTRX-335140 结构式
BCP32121 BTRX-335140 2244614-14-8
BTRX-335140 (CYM-53093) is a potent and selective, orally active κ opioid receptor (KOR) antagonist, has antagonist activity for κOR, μOR and δOR with IC50 values of 0.8 nM, 110 nM, and 6500 nM, respectively. BTRX-335140 endows with favorable in vitro ADMET and in vivo pharmacokinetic profiles and medication-like duration of action in rats.
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