首页   >  
Angiogenesis/Protein Tyrosine Kinase
  >  
Src/Bcr Abl

所有产品分类

所有产品

信号通路

研究领域

天然产物

抗体

多肽

催化剂

杂质对照品

医药中间体

基础原料

Src/Bcr Abl

结构式 货号 产品名称 CAS号
CSF1R-IN-2 结构式
BCP40929 CSF1R-IN-2 2271119-26-5
TPX-0022, also known as CSF1R-IN-2, is an orally bioavailable multi-targeted kinase inhibitor with a novel three-dimensional macrocyclic structure that inhibits the MET, CSF1R (colony stimulating factor 1 receptor) and SRC kinases.
KX2-391 Mesylate 结构式
BCP25173 KX2-391 Mesylate 1080645-95-9
Tirbanibulin, also known as KX-01 and KX2-391, is the first clinical Src inhibitor of the novel peptidomimetic class that targets the peptide substrate site of Src providing more specificity toward Src kinase.
TL02-59 结构式
BCP38228 TL02-59 1315330-17-6
TL02-59 is a novel potent and selective inhibitor of the myeloid Src-family kinase Fgr, suppressing AML cell growth in vitro and in vivo.
DGY-06-116 结构式
BCP37659 DGY-06-116 2556836-50-9
DGY-06-116 is an irreversible covalent, selective Src inhibitor.
PD173955-Analog1 结构式
BCP36116 PD173955-Analog1 185039-99-0
PD 173955-Analog1 is a potent c-Src inhibitor known to have activity against a variety of cancers including colon, lung, head and neck carcinoma.
CH6953755 结构式
BCP35548 CH6953755 2055918-71-1
CH6953755 is a potent, orally active and selective YES1 kinase (a member of the SRC family) inhibitor with an IC50 of 1.8 nM. CH6953755 inhibits YES1 kinase, leading to antitumor activity against YES1 Gene -amplified cancers in vitro and in vivo.
GMB-475 结构式
BCP31499 GMB-475 2490599-18-1
GMB-475 is a degrader of BCR-ABL1 tyrosine kinase based on PROTAC, overcoming BCR-ABL1-dependent drug resistance.
TG 100572 Hydrochloride 结构式
BCP21364 TG 100572 Hydrochloride 867331-64-4
TG 100572 Hydrochloride is a multi-targeted kinase inhibitor which inhibits receptor tyrosine kinases and Src kinases; has IC50s of 2, 7, 2, 16, 13, 5, 0.5, 6, 0.1, 0.4, 1, 0.2 nM for VEGFR1, VEGFR2, FGFR1, FGFR2, PDGFRβ, Fgr, Fyn, Hck, Lck, Lyn, Src, Yes, respectively.
PD 166285 dihydrochloride 结构式
BCP22349 PD 166285 dihydrochloride 212391-63-4
PD-166285 is a potent and broadly active protein tyrosine kinase inhibitor.
pp60c-src Fragment 521-533 结构式
BCP27682 磷酸化 PP60 C-SRC (521-533) 149299-77-4
pp60 c-src (521-533) (phosphorylated) is a peptide corresponding to the pp60c-src carboxy terminal regulatory domain; phosphorylated at Tyr527. Binds to pp60c-src and pp60v-src at the SH2 domain, suppressing their tyrosine kinase activity and transforming potential.
123下一页末页共 81 条记录 1 / 9 页 
2853530911