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Phosphodiesterase/PDE

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Phosphodiesterase/PDE

结构式 货号 产品名称 CAS号
Ro 20-1724 结构式
BCP42971 Ro 20-1724 29925-17-5
Ro 20-1724 is a widely used inhibitor of cyclic nucleotide phosphodiesterase, selective for PDE4 (IC50 = 2.0 μM).
Zaprinast 结构式
BCP38400 扎普司特 37762-06-4
Zaprinast is an inhibitor of the growth of asexual blood-stage malaria parasites (P. falciparum). It acts by inhibiting PfPDE1 and activating GPR35.
HA-155 结构式
BCP37817 HA-155 1229652-22-5
HA-155 is a boronic acid-based compound that inhibits autotaxin (IC50 = 5.7 nM) by selectively binding to its catalytic threonine.
ATX inhibitor 1 结构式
BCP37626 ATX inhibitor 1 2225892-70-4
ATX inhibitor 1 is a potent ATX (IC50=1.23 nM, FS-3 and 2.18 nM, bis-pNPP) inhibitor.
THPP-1 结构式
BCP37557 THPP-1 1257051-63-0
THPP-1 is a potent and orally bioavailable PDE10A inhibitor.
AMG 579 结构式
BCP36114 AMG 579 1227067-61-9
AMG 579 is a potent, selective, and efficacious inhibitor of phosphodiesterase 10A (PDE10A).
Mardepodect hydrochloride 结构式
BCP35070 Mardepodect hydrochloride 2070014-78-5
Mardepodect hydrochloride is a potent, orally active and selective PDE10A inhibitor with an IC50 of 0.37 nM, with >1000-fold selectivity over other PDEs. Mardepodect hydrochloride can cross the blood-brain barrier.
Zatolmilast 结构式
BCP34899 Zatolmilast 1606974-33-7
Zatolmilast(BPN14770) is a phosphodiesterase IV inhibitor.
Deltasonamide 2 结构式
BCP34859 Deltasonamide 2 2088485-34-9
Deltasonamide 2 is a competitive, high affinity PDEδ inhibitor.
PF 04449613 结构式
BCP25929 PF 04449613 1236858-52-8
PF 04449613 is a potent PDE9 inhibitor (IC50 = 22 nM).
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