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GS-9901 Chemical Structure

GS-9901

Data Sheet For research use only. Not for human use.
Cat. No. :BCP44115CAS No. :1640247-87-5Purity:98%
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  • Chemical Properties&Biological Activity
CAS No. 1640247-87-5 Cat. No. BCP44115
Name GS-9901
Synonyms GS 9901; GS9901;
SMILES C1CC1C(C2=NC3=C(C=CC(=C3C(=O)N2C4=CN=CC=C4)Cl)F)NC5=NC(=NC(=C5C#N)N)N
Chemical Name
Formula C22H17ClFN9O M. Wt 477.89
Purity 98% Storage Store at 4-8°C
Description GS-9901 is a potent, orally active and highly selective inhibitor of PI3Kδ (PI3Kdelta IC50 = 1.0nM, HWB delta EC50 = 1.5 nM; CLpr hHep = 0.05 L/h/kg.). GS-9901 displays an excellent pharmacokinetic profile and is efficacious in a rodent model of rheumatoid arthritis. GS-9901 demonstrates efficacy in a rat model of arthritis and is predicted to be suitable for q.d. dosing in humans. The favorable in vitro and in vivo attributes of GS-9901 resulted in its selection as a development candidate.
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