RK-287107 New
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CAS No. | 2171386-10-8 | Cat. No. | BCP30401 |
Name | RK-287107 | ||
Synonyms | RK 287107; RK287107; | ||
SMILES | O=C1NC(N2CCC3(CC2)CN(CCO)C4=C3C(F)=CC(F)=C4)=NC5=C1CCCC5 | ||
Chemical Name | |||
Formula | C22H26F2N4O2 | M. Wt | 416.47 |
Purity | 98% | Storage | Store at 4-8°C |
Description | RK-287107 is a potent TNKS/TNKS2 inhibitor (IC50 = 14.4 nM) with >7000-fold selectivity against the PARP1 enzyme, which inhibits WNT-responsive TCF reporter activity and proliferation of human colorectal cancer cell line COLO-320DM. RK-287107 also demonstrated dose-dependent tumor growth inhibition in a mouse xenograft model. RK-287107 is a promising lead compound for the development of novel tankyrase inhibitors as anticancer agents. |
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