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CXCR

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CXCR

Chemical Structure Cat. No. Product Name CAS No.
USL311 Chemical Structure
BCP33234 USL311 1373268-67-7
USL311 is a selective CXCR4 antagonist, with anti-tumor activity. USL311 prevents the binding of stromal-cell derived factor-1 (SDF-1 or CXCL12) to CXCR4.
Mavorixafor trihydrochloride Chemical Structure
BCP26048 Mavorixafor trihydrochloride 880549-30-4
Mavorixafor is a potent, selective and orally available CXCR4 antagonist, with an IC50 value of 13 nM against CXCR4 125I-SDF binding, and also inhibits the replication of T-tropic HIV-1 (NL4.3 strain) in MT-4 cells and PBMCs with an IC50 of 1 and 9 nM, respectively.
BX471 hydrochloride Chemical Structure
BCP32594 BX471 hydrochloride 288262-96-4
BX471 hydrochloride is a potent, selective non-peptide CCR1 antagonist with Ki of 1 nM for human CCR1, and exhibits 250-fold selectivity for CCR1 over CCR2, CCR5 and CXCR4.
SX-682 Chemical Structure
BCP32154 SX-682 1648843-04-2
SX-682 is a potent and selective Cxcr1/2 inhibitor potentially useful for castration-resistant prostate cancer. CXCR1 and CXCR2 chemokine receptors and their ligands (CXCL1/2/3/7/8) play an important role in tumor progression.
JMS-17-2 Chemical Structure
BCP31312 JMS-17-2 1380392-05-1
JMS-17-2 is a potent and selective antagonist of CX3CR1.
Elubrixin hydrochloride Chemical Structure
BCP23554 Elubrixin hydrochloride 688763-65-7
Elubrixin is a interleukin 8 inhibitor and CXCR2 selective antagonist, which is potentially useful for Inflammatory bowel disease therapies.
Baohuoside I Chemical Structure
BCP30977 Baohuoside I 113558-15-9
Baohuoside I, a flavonoid isolated from Epimedium koreanum Nakai, acts as an inhibitor of CXCR4, downregulates CXCR4 expression, induces apoptosis and shows anti-tumor activity.
ML339 Chemical Structure
BCP30789 ML339 2080300-49-6
ML-339 is a potent and selective hCXCR6 antagonist (IC50 = 140 nM).
MSX-130 Chemical Structure
BCP30792 MSX-130 4051-59-6
MSX-130 is CXCR4 Antagonist.
ATI-2341 Chemical Structure
BCP30749 ATI-2341 1337878-62-2
ATI-2341 is a CXCR4 agonist, induces CXCR4-dependent calcium flux, with an EC50 of 194 nM in CCRF-CEM cells. ATI-2341 is also a potent and efficacious mobilizer of bone marrow hematopoietic cells.
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