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Chemical Structure Cat. No. Product Name CAS No.
GSK2807 Trifluoroacetate Chemical Structure
BCP36148 GSK2807 Trifluoroacetate 2245255-66-5
GSK2807 Trifluoroacetate is a potent, selective and SAM-competitive inhibitor of SMYD3, with a Ki of 14 nM and an IC50 of 130 nM.
AZD-4205 Chemical Structure
BCP36112 AZD-4205 2091134-68-6
AZD4205 is a novel potent and selective janus kinase 1 (JAK1) inhibitor.
SNDX-5613 Chemical Structure
BCP36044 SNDX-5613 2169919-21-3
SNDX-5613 is a potent and specific Menin-MLL inhibitor. It can be used for the research of MLL-rearranged (MLL-r) acute leukemias, including acute lymphoblastic leukemia (ALL) and acute myeloid leukemia (AML).
MI-463 Chemical Structure
BCP36072 MI-463 1628317-18-9
MI-463 is a highly potent and orally bioavailable small molecule inhibitor of the menin-mLL interaction.
MI-538 Chemical Structure
BCP36073 MI-538 1857417-10-7
MI-538 is an inhibitor of the interaction between menin and MLL fusion proteins with an IC50 of 21 nM.
BGP-15 dihydrochloride Chemical Structure
BCP24844 BGP-15 dihydrochloride 66611-37-8
BGP-15 is a PARP inhibitor, with an IC50 and a Ki of 120 and 57 μM, respectively.
GSK620 Chemical Structure
BCP35923 GSK620 2088410-46-0
GSK620 is a novel BD2-selective BET inhibitor in vivo tool , binding to the individual tandem bromodomains [BD1 and BD2] of BRD2, BRD3, BRD4, and BRDT.
GSK046 Chemical Structure
BCP35924 GSK046 2474876-09-8
GSK046 (iBET-BD2) is a selective and orally active inhibitor of BET, with IC50s of 264 nM (BRD2 BD2), 98 nM (BRD3 BD2), 49 nM (BRD4 BD2) and 214 nM (BRDT BD2), respectively.
SP-146 Chemical Structure
BCP35921 SP-146 SP-146
SP-146 is a potent, selective and non-ATP-competitive inhibitor of Aurora B with IC50 of 0.316 nM.
BRD4 Inhibitor-10 Chemical Structure
BCP35872 BRD4 Inhibitor-10 1660117-38-3
BRD4 Inhibitor-10 is a potent and selective BET inhibitor with IC50 of 5 nM and 41 nM for the binding of BRD4-BD1 and BRD4-BD2 to acetylated histones, respectively. BI 894999 is highly selective for BRD2/3/4 and BRDT (Kd of 0.49-1.6 nM), with at least a 200-fold selectivity vs. BRD4-BD1.
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