New Arrivals
| Chemical Structure | Cat. No. | Product Name | CAS No. |
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BCP30845 | N-(p-amylcinnamoyl) Anthranilic Acid New | 110683-10-8 |
N-(p-amylcinnamoyl) Anthranilic Acid (ACA) is a broad spectrum Phospholipase A2 (PLA2) inhibitor and TRP channel blocker. N-(p-amylcinnamoyl) Anthranilic Acid (ACA) is also an effective reversible inhibitor of calcium-activated chloride channels, has potential to treat arrhythmia.
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BCP24252 | Brevianamide F New | 38136-70-8 |
Brevianamide F is a naturally occurring 2,5-diketopiperazine that possess interesting breast cancer resistance protein (BCRP) inhibitory activity.; also shows agonism towards Ca(2+)-channel activity at 100 uM, and has potentiation for use in the treatment of cardiovascular dysfunction.
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BCP28919 | YHO-13351 (free base) New | 912288-64-3 |
YHO-13351 (free base) is the water-soluble prodrug of YHO-13177, which is a potent and specific inhibitor of BCRP.
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BCP28920 | YHO-13351 New | 1346753-00-1 |
YHO-13351 is the water-soluble prodrug of YHO-13177, which is a potent and specific inhibitor of BCRP.
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BCP28921 | Fumitremorgin C New | 118974-02-0 |
Fumitremorgin C is a potent and selective ABCG2/BRCP inhibitor.
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BCP11514 | Lesinurad sodium New | 1151516-14-1 |
Lesinurad sodium is a URAT1 and OAT inhibitor, is determined to be a substrate for the kidney transporters OAT1 and OAT3 with Km values of 0.85 and 2 µM, respectively.
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BCP27717 | Org 25935 hydrochloride New | 949588-40-3 |
Org-25935, also called SCH-900435, is a GlyT-1 inhibitor potentially for the treatment of schizophrenia and alcohol dependence.
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BCP21210 | ALX 5407 New | 571147-18-7 |
ALX 5407 is a potent, selective GlyT1 inhibitor that demonstrates >10-fold greater activity in in vitro functional glycine reuptake assay than racemic (±)-NFPS.
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BCP21322 | Vanoxerine New | 67469-69-6 |
Vanoxerine (GBR12909) is a potent and selective DRI (Dopamine reuptake inhibitor).
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BCP15831 | Tetrabenazine New | 58-46-8 |
Tetrabenazine is a VMAT-inhibitor used for treatment of hyperkinetic movement disorder.
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BCP30846 | Mofezolac New | 78967-07-4 |
Mofezolac, also known as Disopain and N-22, is a cyclooxygenase-1 selective inhibitor used to treat pain, musculoskeletal pain, and arthritis.
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BCP30847 | Verdiperstat New | 890655-80-8 |
Verdiperstat (AZD3241) is a selective, irreversible and orally active myeloperoxidase inhibitor, with an IC50 of 630 nM, and can be used in the research of neurodegenerative brain disorders.
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BCP30848 | JNJ-10229570 New | 524923-88-4 |
JNJ-10229570 is a novel MC1R and MC5R antagonist was used to treat primary human sebaceous cells. It might have a potential for the treatment of acne and other sebaceous gland pathologies.
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BCP30849 | Tyrosine kinase-IN-1 New | 705946-27-6 |
Tyrosine kinase-IN-1 is a multi-targeted tyrosine kinase inhibitor with IC50s of 4, 20, 4, 2 nM for KDR, Flt-1, FGFR1 and PDGFRα, respectively.
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BCP30850 | YF-2 New | 1311423-89-8 |
YF2 is a First-in-Class Histone Acetyltransferase (HAT) Activators for Precision Targeting of Epigenetic Derangements in Lymphoma.
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BCP30851 | Guanabenz New | 5051-62-7 |
Guanabenz is an alpha agonist of the alpha-2 adrenergic receptor that is used as an antihypertensive drug.
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BCP30852 | Radiprodil New | 496054-87-6 |
Radiprodil (RGH-896) is an orally active and selective NMDA NR2B antagonist. A potential therapeutic agent in treatment of neuropathic pain and possibly other chronic pain conditions.
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BCP26187 | CaCCinh-A01 New | 407587-33-1 |
CaCCinh-A01 is an inhibitor of both TMEM16A and calcium-activated chloride channel (CaCC) with IC50s of 2.1 and 10 μM, respectively.
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BCP29329 | Shikonin New | 517-89-5 |
Shikonin is a major component of a Chinese herbal medicine named zicao. Shikonin has shown various biological activities, including inhibition of TNF-α, NF-κB, HIV-1.
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BCP30869 | Sulfalen New | 152-47-6 |
Sulfalene is a long-acting plasma-bound sulfonamide used for respiratory and urinary tract infections and also for malaria.
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