Home   >  
Epigenetics
  >  
Histone Acetyltransferase

Classified by application

All Products

Signaling Pathways

Research Areas

Nature products

Antibodies

Peptides

Catalysts

Impurities

Intermediate

Raw Materials

Histone Acetyltransferase

Chemical Structure Cat. No. Product Name CAS No.
EML 425 Chemical Structure
BCP46797 EML 425 1675821-32-5
EML425 is a potent and selective CREB binding protein (CBP)/p300 inhibitor with IC50s of 2.9 and 1.1 μM, respectively.
L002 Chemical Structure
BCP46453 L002 321695-57-2
L-002 is an inhibitor of p300 histone acyltransferase (KAT3B). L-002 also inhibits acetylation of histones and p53 and suppresses STAT3 activation. In vivo, L-002 potently suppressed tumor growth of TNBC cell line MDA-MB-468 xenografts.
TH 1834 Chemical Structure
BCP45747 TH 1834 2108830-08-4
TH1834 is a novel potent specific histone acetyltransferaseTip60 inhibitor.
TTK21 Chemical Structure
BCP37892 TTK21 709676-56-2
TTK21 is an activator of CBP/p300 histone acetyltransferase activity that activates CBP/p300 histone acetyltransferase activity in a concentration-dependent manner.
P300/CBP-IN-3 Chemical Structure
BCP34907 P300/CBP-IN-3 2299226-01-8
P300/CBP-IN-3, a p300/CBP histone acetyltransferase inhibitor, Compound 6, is sourced from patent WO 2019049061 A1.
GSK4027 Chemical Structure
BCP25140 GSK4027 2079896-25-4
GSK 4027 is a chemical probe for the PCAF/GCN5 bromodomain with an pIC50 of 7.4±0.11 for PCAF in a time-resolved fluorescence resonance energy transfer (TR-FRET) assay.
WM-1119 Chemical Structure
BCP29433 WM-1119 2055397-28-7
WM-1119 is a highly potent, selective inhibitor of lysine acetyltransferase KAT6A with Kd of 2 nM, shows greate bioavailability and specificity for KAT6A than WM-8014.
YF-2 Chemical Structure
BCP30850 YF-2 1311423-89-8
YF2 is a First-in-Class Histone Acetyltransferase (HAT) Activators for Precision Targeting of Epigenetic Derangements in Lymphoma.
NSC228155 Chemical Structure
BCP30383 NSC228155 113104-25-9
NSC228155 is an inhibitor of KIX-KID interaction that acts by enhancing tyrosine phosphorylation of EGFR.
MOZ-IN-2 Chemical Structure
BCP29432 MOZ-IN-2 2055397-88-9
MOZ-IN-2 is an inhibitor of protein MOZ, a member of histone acetyltransferases, with an IC50 of 125 μM.
123下一页共 25 条记录 1 / 3 页 
0086-13720134139