Home   >  
GPCR/G Protein
  >  
CRFR

Classified by application

All Products

Signaling Pathways

Research Areas

Nature products

Antibodies

Peptides

Catalysts

Impurities

Intermediate

Raw Materials

CRFR

Chemical Structure Cat. No. Product Name CAS No.
CP154526 Chemical Structure
BCP26372 CP154526 157286-86-7
CP 154,526 is a selective, non-peptide CRF1 receptor antagonist (Ki values are 2.7 and > 10000 nM for CRF1 and CRF2 receptors respectively).
Verucerfont Chemical Structure
BCP26371 Verucerfont 885220-61-1
Verucerfont is a corticotropin-releasing factor receptor 1 (CRF1) antagonist with IC50s of ~6.1, >1000 and >1000 nM for CRF1, CRF2, and CRF-BP, respectively.
CP 376395 Chemical Structure
BCP28957 CP 376395 175140-00-8
CP-376395 is a CRF1-selective antagonist.
CP 376395 hydrochloride Chemical Structure
BCP28958 CP 376395 hydrochloride 1013933-37-3
CP 376395 hydrochloride is a potent and selective CRF-RI receptor antagonist (Ki value are 12 and >10000 nM for CRF-RI and CRF-RII receptors respectively).
R-121,919 Chemical Structure
BCP23964 R-121,919 195055-03-9
R121919 is a potent small-molecule CRF1 receptor antagonist with a Ki of 2 to 5 nM for the CRF1 receptor and over 1000-fold weaker activity at the CRF2 receptor, CRF-binding protein, or 70 other receptor types.
Pexacerfont Chemical Structure
BCP26369 Pexacerfont 459856-18-9
Pexacerfont is a selective corticotropin-releasing factor (CRF1) receptor antagonist with IC50 of 6.1±0.6 nM for human CRF1 receptor.
0086-13720134139