Home   >  
GPCR/G Protein
  >  
Endothelin Receptor

Classified by application

All Products

Signaling Pathways

Research Areas

Nature products

Antibodies

Peptides

Catalysts

Impurities

Intermediate

Raw Materials

Endothelin Receptor

Chemical Structure Cat. No. Product Name CAS No.
Darusentan Chemical Structure
 BCP13024 Darusentan 171714-84-4
Darusentan (LU-135252; HMR-4005) is an endothelin receptor antagonist.
Hydroxy Bosentan Chemical Structure
 BCP15832 Hydroxy Bosentan 253688-60-7
Hydroxy Bosentan is a metabolite of Bosentan.
Aprocitentan Chemical Structure
 BCP28125 Aprocitentan 1103522-45-7
Aprocitentan is the major and pharmacologically active metabolite of macitentan, which is dual ETA/ETB antagonist designed for tissue targeting.
BQ-123 Chemical Structure
 BCP29354 BQ-123 136553-81-6
BQ-123 is a elective ETA endothelin receptor antagonist (Ki values are 1.4 and 1500 nM at ETA and ETB receptors respectively).
Ro 46-2005 Chemical Structure
 BCP17756 Ro 46-2005 150725-87-4
Ro 46-2005 is a novel synthetic non-peptide endothelin receptor antagonist, inhibits the specific binding of 125I-ET-1 to human vascular smooth muscle cells (ETA receptor) with IC50 of 220 nM.
IRL-1620 Chemical Structure
 BCP09112 IRL-1620 142569-99-1
IRL-1620, also known as SPI-1620, is an endothelin B receptor agonist.
Sitaxsentan sodium Chemical Structure
 BCP08362 Sitaxsentan sodium 210421-74-2
Sitaxsentan sodium (TBC11251 sodium salt) is an orally active, highly selective antagonist of endothelin A receptors.
Ambrisentan Chemical Structure
 BCP22426 Ambrisentan 177036-94-1
Ambrisentan is a selective ET type A receptor (ETAR) antagonist.
Endothelin-1 Acetate Chemical Structure
 BCP27613 Endothelin-1 Acetate 117399-94-7
Endothelin 1 (swine, human) is a synthetic peptide with the sequence of human and swine Endothelin 1, which is a potent endogenous vasoconstrictor. Endothelin 1 acts through two types of receptors ETA and ETB.
Bosentan Chemical Structure
 BCP05202 Bosentan 147536-97-8
Bosentan is a competitive and dual antagonist of endothelin-1 at the endothelin-A (ET-A) and endothelin-B (ET-B) receptors.
12下一页共 16 条记录 1 / 2 页 
0086-15971444841