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Endothelin Receptor

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Endothelin Receptor

Chemical Structure Cat. No. Product Name CAS No.
Sparsentan Chemical Structure
 BCP23969 Sparsentan 254740-64-2
Sparsentan is a highly potent dual angiotensin II and endothelin A receptor antagonist with Kis of 0.8 and 9.3 nM, respectively.
TAK 044 Chemical Structure
 BCP37381 TAK 044 157380-72-8
TAK-044 has been found to be an endothelin receptor antagonist that was once studied against some sort of liver disorders and subarachnoid haemorrhage.
BMS 182874 Hydrochloride Chemical Structure
 BCP33050 BMS 182874 Hydrochloride 1215703-04-0
BMS 182874 hydrochloride is a potent, selective and competitive non-peptide endothelin ETA receptor antagonist (Ki = 48 nM).
BQ-788 Chemical Structure
 BCP29520 BQ-788 173326-37-9
BQ788 is a endothelin B receptor antagonist. BQ788 attenuates stab wound injury-induced reactive astrocytes in rat brain. BQ788 were well tolerated and showed signs of directly and indirectly reducing the viability of melanoma cells.
Carperitide Chemical Structure
 BCP12639 Carperitide 89213-87-6
Carperitide is a polypeptide.
Darusentan Chemical Structure
 BCP13024 Darusentan 171714-84-4
Darusentan (LU-135252; HMR-4005) is an endothelin receptor antagonist.
Hydroxy Bosentan Chemical Structure
 BCP15832 Hydroxy Bosentan 253688-60-7
Hydroxy Bosentan is a metabolite of Bosentan.
Aprocitentan Chemical Structure
 BCP28125 Aprocitentan 1103522-45-7
Aprocitentan is the major and pharmacologically active metabolite of macitentan, which is dual ETA/ETB antagonist designed for tissue targeting.
BQ-123 Chemical Structure
 BCP29354 BQ-123 136553-81-6
BQ-123 is a elective ETA endothelin receptor antagonist (Ki values are 1.4 and 1500 nM at ETA and ETB receptors respectively).
Ro 46-2005 Chemical Structure
 BCP17756 Ro 46-2005 150725-87-4
Ro 46-2005 is a novel synthetic non-peptide endothelin receptor antagonist, inhibits the specific binding of 125I-ET-1 to human vascular smooth muscle cells (ETA receptor) with IC50 of 220 nM.
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