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Nature products
Antibodies
Peptides
Catalysts
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Intermediate
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Raw Materials
Src/Bcr Abl
Chemical Structure | Cat. No. | Product Name | CAS No. |
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BCP38228 | TL02-59 New | 1315330-17-6 |
TL02-59 is a novel potent and selective inhibitor of the myeloid Src-family kinase Fgr, suppressing AML cell growth in vitro and in vivo.
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BCP37659 | DGY-06-116 New | 2556836-50-9 |
DGY-06-116 is an irreversible covalent, selective Src inhibitor.
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BCP36116 | PD173955-Analog1 New | 185039-99-0 |
PD 173955-Analog1 is a potent c-Src inhibitor known to have activity against a variety of cancers including colon, lung, head and neck carcinoma.
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BCP35548 | CH6953755 New | 2055918-71-1 |
CH6953755 is a potent, orally active and selective YES1 kinase (a member of the SRC family) inhibitor with an IC50 of 1.8 nM. CH6953755 inhibits YES1 kinase, leading to antitumor activity against YES1 Gene -amplified cancers in vitro and in vivo.
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BCP31499 | GMB-475 New | GMB-475 |
GMB-475 is a degrader of BCR-ABL1 tyrosine kinase based on PROTAC, overcoming BCR-ABL1-dependent drug resistance.
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BCP21364 | TG 100572 Hydrochloride New | 867331-64-4 |
TG 100572 Hydrochloride is a multi-targeted kinase inhibitor which inhibits receptor tyrosine kinases and Src kinases; has IC50s of 2, 7, 2, 16, 13, 5, 0.5, 6, 0.1, 0.4, 1, 0.2 nM for VEGFR1, VEGFR2, FGFR1, FGFR2, PDGFRβ, Fgr, Fyn, Hck, Lck, Lyn, Src, Yes, respectively.
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BCP22349 | PD 166285 dihydrochloride New | 212391-63-4 |
PD-166285 is a potent and broadly active protein tyrosine kinase inhibitor.
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BCP27682 | pp60c-src Fragment 521-533 New | 149299-77-4 |
pp60 c-src (521-533) (phosphorylated) is a peptide corresponding to the pp60c-src carboxy terminal regulatory domain; phosphorylated at Tyr527. Binds to pp60c-src and pp60v-src at the SH2 domain, suppressing their tyrosine kinase activity and transforming potential.
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BCP30674 | A-770041 New | 869748-10-7 |
A-770041 is selective and orally active Src-family Lck inhibitor; A-770041 is a 147 nM inhibitor of Lck (1 mM ATP) and is 300-fold selective against Fyn, the other Src family kinase involved in T-cell signaling.
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BCP09491 | 1 NM-PP1 New | 221244-14-0 |
1 NM-PP1 is a cell-permeable PP1 analog that acts as a potent and selective inhibitor of mutant kinases over their wild-type progenitors.
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