Home   >  
GPCR/G Protein
  >  
OX Receptor

Classified by application

All Products

Signaling Pathways

Research Areas

Nature products

Antibodies

Peptides

Catalysts

Impurities

Intermediate

Raw Materials

OX Receptor

Chemical Structure Cat. No. Product Name CAS No.
EMPA Chemical Structure
BCP23952 EMPA 680590-49-2
EMPA is a selective antagonist of the OX2 receptor, with 900-fold selectivity in binding for OX2 over OX1.[
SB-334867 Chemical Structure
BCP28004 SB-334867 792173-99-0
SB-334867 free base is a selective non-peptide orexin OX1 receptor antagonist with a pKb value of 7.2.
SB649868 Chemical Structure
BCP28747 SB649868 380899-24-1
SB649868, also known as GSK-649868, is an orexin receptor antagonist potentially for the treatment of insomnia and sleep disorder.
MK4305 Chemical Structure
BCP03512 MK4305 1030377-33-3
Suvorexant (MK-4305) is a potent dual OX receptor antagonist with Ki of 0.55 nM and 0.35 nM for OX1 receptor and OX2 receptor, respectively. Phase 3.
Schisantherin A Chemical Structure
BCP15178 Schisantherin A 58546-56-8
Schisantherin A is a dibenzocyclooctadiene lignan isolated from the fruit of Schisandra sphenanthera. Schisantherin A inhibits p65-NF-κB translocation into the nucleus by IκBα degradation.
TCS 1102 Chemical Structure
BCP08369 TCS 1102 916141-36-1
TCS 1102 is a potent, dual orexin receptor antagonist (Ki values are 0.2 and 3 nM for OX2 and OX1 receptors respectively).
MK-3697 Chemical Structure
BCP08557 MK-3697 1224846-01-8
MK-3697 is a potent and selective Orexin receptor antagonist with Ki = 0.95 nM.
MK6096 Chemical Structure
BCP07891 MK6096 1088991-73-4
MK-6096 is an orally bioavailable potent and selective reversible antagonist of Orexin 1 Receptor (OX(1)R) and Orexin 2 Receptor (OX(2)R).
MK1064 Chemical Structure
BCP19608 MK1064 1207253-08-4
MK-1064 is a selective orexin 2 receptor antagonist (2-SORA) for the research of insomnia.
SB408124 Chemical Structure
BCP02343 SB408124 288150-92-5
SB-408124 (SB 408124)is a selective non-peptide orexin OX1 receptor antagonist .
12下一页共 17 条记录 1 / 2 页 
0086-13720134139