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Histamine Receptor

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Histamine Receptor

Chemical Structure Cat. No. Product Name CAS No.
Thioperamide Chemical Structure
 BCP39480 Thioperamide 106243-16-7
Thioperamide is a potent histamine H3 and H4 antagonist/inverse agonist (Ki = 25 and 27 nM for human recombinant H3 and H4 receptors, respectively). Thioperamide can cross the blood-brain barrier freely.
Thioperamide maleate Chemical Structure
 BCP39479 Thioperamide maleate 148440-81-7
Thioperamide maleate is a selective histamine H3 receptor antagonist that crosses the blood-brain barrier.
JNJ-5207852 Chemical Structure
 BCP37369 JNJ-5207852 398473-34-2
JNJ-5207852 is a selective and potent histamine H3 receptor (H3R) antagonist, with pKis of 8.9, 9.24 for rat and human H3R, respectively.
Thonzylamine Chemical Structure
 BCP25799 Thonzylamine 91-85-0
Thonzylamine is a first-generation ethylenediamine H1-antihistamine.
Doxepin-d3 Hydrochloride Chemical Structure
 BCP33258 Doxepin-d3 Hydrochloride 347840-07-7
Doxepin D3 Hydrochloride is a deuterium labeled Doxepin Hydrochloride.Doxepin is a tricyclic antidepressant (TCA) used for the treatment of major depression and anxiety.
Clobenpropit dihydrobromide Chemical Structure
 BCP33039 Clobenpropit dihydrobromide 145231-35-2
Clobenpropit dihydrobromide is an extremely potent histamine H3 antagonist/inverse agonist (pA2=9.93). Also displays partial agonist activity at H4 receptors; induces eosinophil shape change with an EC50 of 3 nM.
LML134 Chemical Structure
 BCP32719 LML134 1542135-76-1
LML134 is an orally active and high selective Histamine 3 receptor (H3R) inverse agonist with Kis of 0.3 nM and 12 nM for hH3R cAMP and hH3R bdg.
Imetit Dihydrobromide Chemical Structure
 BCP31622 Imetit Dihydrobromide 32385-58-3
Imetit Dihydrobromide is a histamine H3 receptor (H3R) agonist.
Metiamide Chemical Structure
 BCP21503 Metiamide 34839-70-8
Metiamide is a histamine H2-receptor antagonist developed from another H2 antagonist, burimamide.
Pemirolast potassium Chemical Structure
 BCP21138 Pemirolast potassium 100299-08-9
Pemirolast potassium is a potent histamine H1 antagonist and mast cell stabilizer that acts as an antiallergic agent. It has also been studied for the treatment of asthma. Pemirolast potently attenuates paclitaxel hypersensitivity reactions through inhibition of the release of sensory neuropeptides in rats. Pemirolast reduces cisplatin-induced kaolin intake in rats.
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