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Histone Methyltransferase

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Histone Methyltransferase

Chemical Structure Cat. No. Product Name CAS No.
GSK3368715 dihydrochloride Chemical Structure
 BCP38359 GSK3368715 dihydrochloride 1628925-77-8
GSK3368715 dihydrochloride is a novel potent type-I protein arginine methyltransferases (PRMTs) inhibitor.
LEM-14 Chemical Structure
 BCP38013 LEM-14 1814881-70-3
LEM-14 is a specific NSD2 inhibitor.
TM2-115 Chemical Structure
 BCP38007 TM2-115 1197196-47-6
TM2-115 is a potent histone methyltransferase inhibitor with rapid antimalarial activity against all blood stage forms in Plasmodium falciparum
A-196 Chemical Structure
 BCP37560 A-196 1982372-88-2
A 196 is a potent and selective inhibitor of SUV420H1/H2 (IC50 = 25 and 144 nM, respectively) with 100-fold selectivity over other histone methyltransferases and non-epigenetic targets. It was shown to inhibit the di- and tri-methylation of H4K20me in multiple cell lines (IC50 < 1 μM).
Ezh2-IN-2 Chemical Structure
 BCP37576 Ezh2-IN-2 2238821-31-1
EZH2-​IN-​2 is a EZH2 inhibitor.
BAY-598 Chemical Structure
 BCP37130 BAY-598 1906919-67-2
BAY-598 is selective small molecule inhibitor of SMYD2 with an IC50 of 27 nM.
CPI-1612 Chemical Structure
 BCP36917 CPI-1612 2374971-81-8
CPI-1612 is an orally bioavailable EP300/CBP histone acetyltransferase inhibitor
CPI 169 R-enantiomer Chemical Structure
 BCP36903 CPI 169 R-enantiomer 1802175-07-0
CPI 169 R-enantiomer is a novel and potent EZH2 inhibitor.
MS1943 Chemical Structure
 BCP36892 MS1943 2225938-17-8
MS1943 is a first-in-class, orally bioavailable EZH2 selective degrader. It significantly reduces EZH2 protein levels in numerous triple-negative breast cancer (TNBC) and other cancer and noncancerous cell lines. MS1943 effectively blocks proliferation of multiple TNBC and other cancer cell lines.
EPZ004777 HCl Chemical Structure
 BCP36786 EPZ004777 HCl 1380316-03-9
EPZ004777 hydrochloride is the hydrochloride salt of EPZ004777, which is a potent, selective DOT1L inhibitor with IC50 of 0.4 nM.
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