Classified by application
All Products
Signaling Pathways
- Angiogenesis/Protein Tyrosine Kinase
- Apoptosis Pathway
- Cell Cycle/DNA Damage
- Epigenetics
-
GPCR/G Protein
- Melatonin Receptor
- Urotensin Receptor
- Neurotensin Receptor
- Motilin Receptor
- Glucose Transporter
- Adenylate Cyclase
- Cholecystokinin Receptor
- TGR5
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- Imidazoline Receptor
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- Sigma Receptor
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- OX Receptor
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- NK Receptor
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- mAChR
- P2 Receptor
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- Smoothened/Smo
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- Hormone Pathay
- Ion Channel/Membrane Transporter
- Jak/Stat Pathway
- MAPK Pathway
- Microbiology/Virology
-
Neuro Signaling Pathway
- Imidazoline Receptor
- Monoamine Oxidase
- COMT
- Amyloid β
- NK Receptor
- Beta secretase
- AChE
- SSRI
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- P glycoprotein
- Opioid Receptor
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- mGluR
- Histamine Receptor
- Gamma secretase
- Dopamine Transporter
- 5 HT Receptor/Serotonin Receptor
- FAAH
- P2 Receptor
- nAChR
- CGRP Receptor
- COX
- GABA Receptor
- mAChR
- NFκB
- PI3K/Akt/mTOR
-
Protease/Metabolic Enzyme
- 11β HSD
- COMT
- Carboxypeptidase
- ACC
- Xanthine Oxidase
- Mitochondrial Metabolism
- Pyruvate Kinase
- SCD
- ALDH
- Serine Protease
- Neprilysin
- CETP
- FTase
- MLR
- MAGL
- Carbonic Anhydrase
- E1 E2 E3 Enzyme
- Elastase
- Glucokinase
- ROR
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- PAI1
- Aldose Reductase
- Tyrosinase
- FAS
- DGAT
- Lipoxygenase
- Nampt
- IDO
- IDH
- MMP
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- Phosphatase
- Thrombin
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- RAR/RXR
- HMGCR
- FAAH
- Gamma secretase
- RAAS/ACE
- Caspase
- HIV Protease
- Aminopeptidase
- HCV Protease
- HSP
- Tryptophan Hydroxylase/TPH
- Factor Xa
- DPP
- Procollagen C Proteinase
- Integrase
- Phosphodiesterase/PDE
- Phospholipase
- LXR
- Proteasome
- Cytochrome P450
- TGF beta/Smad
- Wnt/Stem Cell
- Others Pathway
Research Areas
- Metabolic Disease
- Neurological Disease
- Endocrinology
- Diabetes
- Cardiovascular Disease
- Immunology
- Allergy
- Inflammation
- Infection
- Cancer
Nature products
Antibodies
Peptides
Catalysts
Impurities
Intermediate
- Amino acid
- Ammonia Series
- Nucleoside Series
- Azaindazole
- Pyridazine Series
- Quinazoline
- Pyrimidine Series
- Pyrazole Series
- Quinoline Series
- Boric acid
- Pyrrole Series
- Thiophene Series
- Saccharide
- Azaindole
- Indole Series
- Piperidine Series
- Indazole Series
- Heterocyclic Series
- Pyridine Series
- Benzene Series
Raw Materials
Histone Methyltransferase
Chemical Structure | Cat. No. | Product Name | CAS No. |
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BCP38359 | GSK3368715 dihydrochloride New | 1628925-77-8 |
GSK3368715 dihydrochloride is a novel potent type-I protein arginine methyltransferases (PRMTs) inhibitor.
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BCP38013 | LEM-14 New | 1814881-70-3 |
LEM-14 is a specific NSD2 inhibitor.
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BCP38007 | TM2-115 New | 1197196-47-6 |
TM2-115 is a potent histone methyltransferase inhibitor with rapid antimalarial activity against all blood stage forms in Plasmodium falciparum
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BCP37560 | A-196 New | 1982372-88-2 |
A 196 is a potent and selective inhibitor of SUV420H1/H2 (IC50 = 25 and 144 nM, respectively) with 100-fold selectivity over other histone methyltransferases and non-epigenetic targets. It was shown to inhibit the di- and tri-methylation of H4K20me in multiple cell lines (IC50 < 1 μM).
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BCP37576 | Ezh2-IN-2 New | 2238821-31-1 |
EZH2-IN-2 is a EZH2 inhibitor.
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BCP37130 | BAY-598 New | 1906919-67-2 |
BAY-598 is selective small molecule inhibitor of SMYD2 with an IC50 of 27 nM.
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BCP36917 | CPI-1612 New | 2374971-81-8 |
CPI-1612 is an orally bioavailable EP300/CBP histone acetyltransferase inhibitor
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BCP36903 | CPI 169 R-enantiomer New | 1802175-07-0 |
CPI 169 R-enantiomer is a novel and potent EZH2 inhibitor.
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BCP36892 | MS1943 New | 2225938-17-8 |
MS1943 is a first-in-class, orally bioavailable EZH2 selective degrader. It significantly reduces EZH2 protein levels in numerous triple-negative breast cancer (TNBC) and other cancer and noncancerous cell lines. MS1943 effectively blocks proliferation of multiple TNBC and other cancer cell lines.
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BCP36786 | EPZ004777 HCl New | 1380316-03-9 |
EPZ004777 hydrochloride is the hydrochloride salt of EPZ004777, which is a potent, selective DOT1L inhibitor with IC50 of 0.4 nM.
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