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GPR

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GPR

Chemical Structure Cat. No. Product Name CAS No.
AMG-837 calcium hydrate Chemical Structure
 BCP28243 AMG-837 calcium hydrate 1259389-38-2
AMG 837 calcium hydrate is a potent GPR40 agonist(EC50=13 nM) with a superior pharmacokinetic profile and robust glucose-dependent stimulation of insulin secretion in rodents.
AF64394 Chemical Structure
 BCP29864 AF64394 1637300-25-4
AF64394 is a GPR3 inverse agonist, with a pIC50 of 7.3.
MS21570 Chemical Structure
 BCP29503 MS21570 65373-29-7
MS21570 is a GPR171 antagonist that reduces anxiety-like behavior and fear conditioning in mice.
TC-O 9311 Chemical Structure
 BCP28396 TC-O 9311 444932-31-4
TC-O9311 is a potent GPR139 agonist (EC50 = 39 nM in CHO-K1 cells expressing human GPR139).
LY-2881835 Chemical Structure
 BCP28854 LY-2881835 1292290-38-0
LY2881835 is a potent and selective GPR40 agonist potentially for treatment of type 2 diabetes mellitus.
FTBMT Chemical Structure
 BCP29255 FTBMT 1358575-02-6
FTBMT is a selective GPR52 agonist. It demonstrates antipsychotic-like and procognitive effects in rodents and has revealed a potential therapeutic agent for schizophrenia.
AM-1638 Chemical Structure
 BCP13218 AM-1638 1142214-62-7
AM-1638 is a potent and orally Bioavailable GPR40/FFA1 Full Agonist.
CID16020046 Chemical Structure
 BCP20242 CID16020046 834903-43-4
CID 16020046 is a potent and selective GPR55(LPI receptor) antagonist; inhibitsGPR55 constitutive activity with IC50 of 0.15 uM.
AMG 837 Chemical Structure
 BCP14587 AMG 837 865231-46-5
AMG 837 is a potent GPR40 agonist(EC50=13 nM) with a superior pharmacokinetic profile and robust glucose-dependent stimulation of insulin secretion in rodents.
GTPL5846 Chemical Structure
 BCP14892 GTPL5846 83797-69-7
6-OAU(GTPL5846; 6-n-octylaminouracil) is a surrogate agonist of GPR84; activates human GPR84 in the presence of Gqi5 chimera in HEK293 cells with an EC50 of 105 nM in the PI assay.
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