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Signaling Pathways
- Angiogenesis/Protein Tyrosine Kinase
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- Epigenetics
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GPCR/G Protein
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Neuro Signaling Pathway
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Protease/Metabolic Enzyme
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Research Areas
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Nature products
Antibodies
Peptides
Catalysts
Impurities
Intermediate
- Amino acid
- Ammonia Series
- Azaindazole
- Pyridazine Series
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- Nucleoside Series
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- Boric acid
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- Saccharide
- Azaindole
- Indole Series
- Piperidine Series
- Indazole Series
- Heterocyclic Series
- Benzene Series
- Pyridine Series
Raw Materials
Histone Demethylase
Chemical Structure | Cat. No. | Product Name | CAS No. |
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BCP37630 | KDM5-IN-1 New | 1628210-26-3 |
KDM5-IN-1 is a potent, selective and orally bioavailable KDM5 inhibitor.
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BCP37627 | KDM5-C70 New | 1596348-32-1 |
KDM5-C70 is a JARID1 Histone Demethylases Inhibitor. KDM5-C70 had an antiproliferative effect in myeloma cells, leading to genome-wide elevation of H3K4me3 levels.
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BCP33218 | CC-90011 besylate New | 2097523-60-7 |
CC-90011 is a potent and orally active LSD1 inhibitor. CC-90011 binds to and inhibits LSD1, a demethylase that suppresses the expression of target genes by converting the di- and mono-methylated forms of lysine at position 4 of histone H3 (H3K4) to mono- and unmethylated H3K4, respectively.
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BCP25948 | OG-L002 hydrochloride New | 1357298-75-9 |
OG-L002 HCl is an inhibitor of LSD1.
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BCP32624 | KDM4D-IN-1 New | 2098902-68-0 |
KDM4D-IN-1 is a new histone lysine demethylase 4D (KDM4D) inhibitor with an IC50 value of 0.41±0.03 μM.
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BCP31703 | KDOAM-25 New | 2230731-99-2 |
KDOAM-25 is a potent and highly selective KDM5 sub-family of histone lysine demethylases inhibitor with IC50s of 71 nM, 19 nM, 69 nM, 69 nM for KDM5A, KDM5B, KDM5C, KDM5D, respectively. KDOAM-25 increases global H3K4 methylation at transcriptional start sites and impairs proliferation in multiple myeloma MM1S cells.
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BCP30840 | GSK-467 New | 1628332-52-4 |
GSK467 is a potent and selective inhibitor of KDM5 (also known as JARID1). GSK467 exploits unique binding modes.
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BCP30535 | T-3775440 New | 1422620-34-5 |
T-3775440 is a novel potent, selecitve, irreversible LSD1 inhibitor with IC50 of 2.1 nM.
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BCP30534 | T-3775440 hydrochloride New | 1422535-52-1 |
T-3775440 hydrochloride is a potent, selecitve, irreversible LSD1 inhibitor.
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BCP30529 | Corin New | 1808113-09-8 |
Corin is a dual inhibitor of histone lysine specific demethylase (LSD1) and histone deacetylase (HDAC), with a Ki(inact) of 110 nM for LSD1 and an IC50 of 147 nM for HDAC1.
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