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Casein Kinase

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Casein Kinase

Chemical Structure Cat. No. Product Name CAS No.
Longdaysin Chemical Structure
BCP32583 Longdaysin 1353867-91-0
Longdaysin is a novel inhibitor of CK1, ERK2, and CDK7 kinases.
BioE-1115 Chemical Structure
BCP32544 BioE-1115 1268863-35-9
BioE-1115 is a highly selective and potent PAS kinase (PASK) inhibitor with an IC50 of ~4 nM. BioE-1115 is also a potent casein kinase 2α inhibitor with an IC50 of ~10 μM.
TMCB Chemical Structure
BCP27716 TMCB 905105-89-7
TMCB is a dual-kinase inhibitor. It acts by inhibiting both casein kinase 2 (CK2) and extracellular-signal-regulated kinase 8 (ERK8).
NCC007 Chemical Structure
BCP30832 NCC007 NCC007
NCC007 is a novel CKIα and CKIδ dual inhibitor.
PF-5006739 Chemical Structure
BCP29752 PF-5006739 1293395-67-1
PF-5006739 is a potent casesin kinase 1δ/ε inhibitor (IC50 values are 3.9 and 17 nM, respectively). Mediates circadian rhythm phase-delaying effects in vivo. Attenuates opioid drug seeking behaviour in addiction in vivo models.
PF4800567 Chemical Structure
BCP28458 PF4800567 1188296-52-7
PF-4800567 is a selective inhibitor of casein kinase 1ε (CK1ε; IC50 = 32 nM) with greater than 20-fold selectivity over CK1δ.
TA-01 Chemical Structure
BCP24229 TA-01 1784751-18-3
TA-01 is a potent CK1 and p38 MAPK inhibitor, with IC50s of 6.4 nM, 6.8 nM, 6.7 nM for CK1ε, CK1δ and p38 MAPK, respectively.
Ellagic acid Chemical Structure
BCP10830 Ellagic acid 476-66-4
Ellagic acid is a natural antioxidant, and acts as a potent and ATP-competitive CK2 inhibitor, with an IC50 of 40 nM and a Ki of 20 nM.
IC 261 Chemical Structure
BCP16652 IC 261 186611-52-9
IC261 is a reversible, ATP-competitive inhibitor of casein kinase 1 (CK1) that inhibits Ckiδ and Ckiε (IC50 = ~1 μM for both), as well as CK1α (IC50 = 16 μM).
SR-3029 Chemical Structure
BCP20656 SR-3029 1454585-06-8
SR-3029 is a potent and selective casein kinase 1δ/1ε (CK1δ/ε) inhibitor with potent antiproliferative properties SR-3029 shoed IC50:= 97 nM in MTT assays against the human A375 melanoma cell line and have physical, in vitro and in vivo PK properties suitable for use in proof of principle animal xenograft studies against human cancer cell lines.
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