Home   >  
Epigenetics
  >  
Epigenetic Reader Domain

Classified by application

All Products

Signaling Pathways

Research Areas

Nature products

Antibodies

Peptides

Catalysts

Impurities

Intermediate

Raw Materials

Epigenetic Reader Domain

Chemical Structure Cat. No. Product Name CAS No.
A1874 Chemical Structure
 BCP32647 A1874 2064292-12-0
A1874 is a nutlin-based and BRD4-degrading PROTAC which induces BRD4 degradation in cells.
dBET57 Chemical Structure
 BCP32540 dBET57 1883863-52-2
dBET57 is a novel BRD4 heterobifunctional small-molecule ligand (PROTAC) which exhibits significant and selective degradation of BRD4 BD1 but is inactive on BRD4 BD2.
(R)-JQ-1 (carboxylic acid) Chemical Structure
 BCP32538 (R)-JQ-1 (carboxylic acid) 202592-24-3
JQ1 Carboxylic Acid, also known as JQ1 Acid, is an inhibitor of bromodomain and extra terminal domain (BET) family proteins.
QCA570 Chemical Structure
 BCP32101 QCA570 2207569-08-0
QCA570 is a potent BET degrader based on PROTAC, with an IC50 of 10 nM for BRD4 BD1 Protein.
OXFBD04 Chemical Structure
 BCP31554 OXFBD04 OXFBD04
OXFBD04 shows improved BRD4(1) affinity (IC50 = 166 nM), optimised physicochemical properties (LE = 0.43; LLE = 5.74; SFI = 5.96), and greater metabolic stability (t½ = 388 min).
CBP-IN-1 Chemical Structure
 BCP31464 CBP-IN-1 2222941-37-7
CBP-IN-1 is a potent p300/CBP bromodomain inhibitor.
MZ 1 Chemical Structure
 BCP31482 MZ 1 1797406-69-9
MZ1 is a potent inducer of reversible, long-lasting and selective removal of BRD4 over BRD2 and BRD3.
GSK4027 Chemical Structure
 BCP25140 GSK4027 2079896-25-4
GSK 4027 is a chemical probe for the PCAF/GCN5 bromodomain with an pIC50 of 7.4±0.11 for PCAF in a time-resolved fluorescence resonance energy transfer (TR-FRET) assay.
E-7386 Chemical Structure
 BCP30544 E-7386 1799824-08-0
E-7386 is an orally active CBP/beta-catenin modulator.
INCB054329 Racemate Chemical Structure
 BCP30528 INCB054329 Racemate 1628607-62-4
INCB054329 Racemate is a BET protein inhibitor.
123下一页末页共 95 条记录 1 / 10 页 
0086-15971444841