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PKA

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PKA

Chemical Structure Cat. No. Product Name CAS No.
Fasudil Chemical Structure
BCP26821 Fasudil 103745-39-7
Fasudil, a Rho-kinase inhibitor, has been shown to reduce portal venous pressure in cirrhotic rats.
Fasudil hydrochloride Chemical Structure
BCP26351 Fasudil hydrochloride 105628-07-7
Fasudil Hydrochloride is a potent inhibitor of ROCK1, PKA, PKC, and MLCK with Kis of 0.33 μM, 1.0 μM, 9.3 μM and 55 μM, respectively.
Dibutyryl adenosine cyclophosphate calcium Chemical Structure
BCP23536 Dibutyryl adenosine cyclophosphate calcium 938448-87-4
Bucladesine calcium salt(DC2797 calcium salt) is a membrane permeable selective activator of PKA.
CCG215022 Chemical Structure
BCP18562 CCG215022 1813527-81-9
CCG215022 is a potent GRK2 and GRK5 inhibitor. CCG215022 exhibited nanomolar IC50 values against both GRK2 and GRK5 and good selectivity against other closely related kinases such as GRK1 and PKA.
AT13148 Chemical Structure
BCP08961 AT13148 1056901-62-2
AT13148 is a novel oral multi-AGC kinase inhibitor with potent pharmacodynamic and antitumor activity
AT7867 Chemical Structure
BCP02406 AT7867 857531-00-1
AT7867 is a potent ATP-competitive inhibitor of Akt1/2/3 and p70S6K/PKA with IC50 of 32 nM/17 nM/47 nM and 85 nM/20 nM, respectively; little activity outside the AGC kinase family.
H-89 Chemical Structure
BCP02706 H-89 127243-85-0
H 89 2HCl is a potent PKA inhibitor with Ki of 48 nM, 10-fold selective for PKA than PKG, greater than 500-fold selectivity than PKC, MLCK, calmodulin kinase II and casein kinase I/II.
H-89 dihydrochloride hydrate Chemical Structure
BCP15626 H-89 dihydrochloride hydrate 130964-39-5
H-89 (dihydrochloride) is a potent inhibitor of cyclic AMP-dependent protein kinase (protein kinase A) with IC50 of 48 nM and has weak inhibition on PKG, PKC, Casein Kinase, and others kinases.
Staurosporine Chemical Structure
BCP27724 Staurosporine 62996-74-1
Staurosporine is a very potent universal inhibitor of protein kinases but showing little selectivity, with IC50 of 6 nM, 15 nM, 2 nM, and 3 nM for PKC, PKA, c-Fgr, and Phosphorylase kinase, respectively.
Bucladesine Chemical Structure
BCP09391 Bucladesine 16980-89-5
Bucladesine is a membrane permeable selective activator of PKA.
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