GSK2798745 New
Data Sheet
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| CAS No. | 1419609-94-1 | Cat. No. | BCP38659 |
| Name | GSK2798745 | ||
| Synonyms | GSK-2798745; GSK 2798745; | ||
| SMILES | CC1(CCCC2(C1)CN(C(=O)O2)C3=NC=C(N=C3)C(C)(C)O)CN4C=NC5=C4C=C(C=C5)C#N | ||
| Chemical Name | |||
| Formula | C25H28N6O3 | M. Wt | 460.53 |
| Purity | 98% | Storage | Store at 4-8°C |
| Description | GSK2798745 is a potent and selective TRPV4 Ion Channel Inhibitor with IC50 = 1.8 nM. GSK2798745 is potentially useful for the treatment of pulmonary edema associated with congestive heart failure. GSK2798745 demonstrated efficacy in an in vivo rat PK/PD model of pulmonary edema, excellent TRP selectivity (M5, A1, C3, and C6 > 25 μM), and an adequate preclinical safety profile that enabled its candidate selection and subsequent progression to clinical trials. | ||
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